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N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(butan-2-yl)[2-methyl-2-(morpholin-4-ylmethyl)propyl](pyridin-4-ylmethyl)amine
1-(3,4-dimethylphenyl)-N-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(3-methylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2R)-2-({2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazol-4-yl}formamido)propanamide
N'-cyclopentyl-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]butanediamide
4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
(2S,4S)-N-ethyl-4-(4-{2-[(4-fluorophenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
(1R,3s,6r,8S)-4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-azatricyclo[4.3.1.13,8]undecane
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(pyridin-2-ylmethyl)piperazine
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2-[3-(trifluoromethyl)phenyl]acetamide
3-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}propanamide
6-methyl-2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}pyridine-3-carbonitrile
(2S,4R)-4-amino-N,N-diethyl-1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]pyrrolidine-2-carboxamide
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
ethyl 4-(2-oxo-1-phenylpyrrolidine-3-carbonyl)piperazine-1-carboxylate
1-{[4-(3-benzyl-1H-1,2,4-triazol-5-yl)phenyl]methyl}-1H-1,2,3,4-tetrazole
1-(furan-2-carbonyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,4-diazepane
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanamide
2,2-dimethyl-N-{1-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
4-ethyl-3-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aR,8aR)-7-[6-(4-fluorophenyl)pyridazin-3-yl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
3-[({1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
4-(2-benzyl-1,3-benzoxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[1-(1-benzofuran-2-carbonyl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
1-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
2-(3-fluorophenyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
1,5-dimethyl-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1H-indazole
5-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]piperidin-2-one
1-(2-{2-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)imidazolidin-2-one
N-(pyrimidin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-chloro-4-{[1-(cyclobutylmethyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclobutanecarboxamide
5-(2-butoxy-4-fluorophenyl)-1-methyl-1H-1,2,3,4-tetrazole
1-(1-cyclopentanecarbonylpiperidin-4-yl)-3-(2-fluoro-4-methylphenyl)urea
5-benzyl-2-methyl-4-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]pyrimidine
({4-ethyl-5-[1-(quinoxalin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
7-fluoro-2-methyl-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]quinoline-4-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(2-phenylethyl)piperidine-3-carboxamide
2-{1-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-imidazol-2-yl}quinoline
N-[(3-chlorophenyl)methyl]-N-cyclopropylpyridazine-3-carboxamide
4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2-methyl-1-(propan-2-yl)piperazine
2-ethyl-5-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}pyrimidine
N-(1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}pyrrolidin-3-yl)-N-ethylacetamide
5-{2-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
methyl 4-[4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]benzoate
2-tert-butyl-N-[(3-methoxyphenyl)methyl]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-amine
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
2-[methyl(pyridin-2-ylmethyl)amino]-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide