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methyl 5-cyano-2-methyl-6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyridine-3-carboxylate
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]benzamide
[(2S,6S)-4-[2-(2-ethoxyphenoxy)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-[(2,3-dimethoxyphenyl)methyl]-5-[1-(4-methoxyphenyl)-1H-pyrazol-3-yl]-4-methyl-1,3-thiazol-2-amine
4-{[2-(3-chloro-4-hydroxyphenyl)-1H-imidazol-1-yl]methyl}benzoic acid
1-(furan-3-ylmethyl)-1-methyl-3-{5-[(4-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
(3aS,6aS)-2-cyclopentyl-5-(thian-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
({4-ethyl-5-[1-(4-fluoro-2-methylbenzoyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
8-(1,3-benzothiazol-2-ylmethyl)-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[4-(4-fluorophenyl)oxan-4-yl]-1-methyl-1H-1,2,4-triazole
4-(propan-2-yl)-6-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidin-2-amine
1-{9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
3-(azocan-1-ylmethyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1'-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
2-(5-methoxy-1,3-benzoxazol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-{4-hydroxy-1-[(3-methylphenyl)methyl]piperidin-4-yl}-N-(4-methoxyphenyl)-1-benzofuran-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-ethoxyethyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(3-fluorophenyl)methyl]-1H-pyrazole-4-carboxamide
2-(1,2-benzoxazol-3-yl)-1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
2-{[(2,3-difluorophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(pyridin-4-yl)propanamide
2-(3-hydroxypropyl)-8-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
ethyl 5-(2-methylpropanoyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{1-[(3-chloro-5-fluorophenyl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
N-({3-methyl-7-[4-(2-methylpropyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(pyrimidin-2-ylsulfanyl)acetamide
methyl 4-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperazine-1-carboxylate
N-(2,3-dimethylphenyl)-N'-[2-(3-hydroxypiperidin-1-yl)ethyl]propanediamide
N-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
N-[(4-methylphenyl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
8-acetyl-2-[(2-chloro-4-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2,3-dimethyl-7-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
ethyl 4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-[(5-methylpyrazin-2-yl)methyl]-8-(5-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-3-(2-methoxyphenyl)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
8-{[3-(cyclopentyloxy)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-[(3-methylphenyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(dimethylamino)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)benzamide
2-[(2-fluorophenyl)methyl]-6-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,3-benzoxazole
3-({3-tert-butyl-1-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-methyl-1'-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(3R,4S)-1-cyclopentyl-4-(3-methoxyphenyl)pyrrolidin-3-amine
1-{2-[(4aS,8aR)-1-(2-methylpropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
[4-({1-[(2-cyclohexylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
2-(3-methoxypropyl)-8-[3-(thiophen-3-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
4-[3-(cyclohexyloxy)-2-hydroxypropyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-cyclopropanecarbonyl-4-(thiophen-2-ylmethyl)-1,4-diazepane-6-carboxylic acid
3-cyclopropyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1H-pyrazole-5-carboxamide