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N-cycloheptyl-1-(2-ethoxyethyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)[(2-methoxyphenyl)methyl]methylamine
N-ethyl-2-[2-(1H-pyrazol-1-yl)butanamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
(3aS,6aS)-5-(4-cyclopentylpyrimidin-2-yl)-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3R,4S)-1-(4-chloro-2-fluorobenzoyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-2-(thianthren-1-yl)acetic acid
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]ethan-1-one
1-{1-[2-(propan-2-yloxy)acetyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
ethyl 2-amino-3-cyano-4-[5-(hydroxymethyl)furan-2-yl]-5,6,7,8-tetrahydroquinoline-6-carboxylate
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
(3S,5R)-5-(pyrrolidine-1-carbonyl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidine-3-carboxylic acid
9-[(5-methylthiophen-2-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(3-chloropyridin-2-yl)piperazine-1-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane
2-(2-hydroxyethyl)-9-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepan-6-ol
6-(1-phenylcyclohexanecarbonyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}but-3-enamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-cyclopropylacetamide
4-({[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl](methyl)amino}methyl)-1-ethylpyrrolidin-2-one
methyl 5-{[(3,5-difluorophenyl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,6S)-3-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-9-methyl-3,9-diazabicyclo[4.2.1]nonane
[(3R,4R)-1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
[3-(3-methylbut-2-en-1-yl)-1-(pyridin-2-ylmethyl)piperidin-3-yl]methanol
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
5-(4-methoxyphenyl)-3-[4-(4-methoxyphenyl)piperazin-1-yl]-1,2,4-triazine
(3S,4S)-1-[(2-hydroxy-5-methylphenyl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetamide
3-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]propanamide
5-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-1,3-oxazole
(1R,5R)-6-[(2E)-2-methylbut-2-en-1-yl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
prop-2-en-1-yl N-methyl-N-({1-[(3S,5S)-5-(methylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)carbamate
2-[(4aR,7aS)-4-(1-methyl-1H-pyrazole-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
4-cyclopropyl-6-[3-(1H-pyrazol-5-yl)phenyl]pyrimidine
(3S,4R)-3-methoxy-1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]piperidin-4-amine
{1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
methyl (1R,3S,3aR,6aS)-1-ethyl-3-(4-hydroxyphenyl)-4,6-dioxo-5-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
8-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
9-(oxolane-2-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-aminoethyl)-N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-1H-1,2,3-triazole-4-carboxamide
4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-N-(4-fluorophenyl)piperazine-2-carboxamide
2-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-1,3-thiazole-4-carboxamide
N-{2-methyl-1-[7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}furan-3-carboxamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-[(4R)-2-oxo-1,3-thiazolidine-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2-chloro-6-fluorophenyl)-N-[2-(oxan-2-yl)ethyl]acetamide
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one