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N-{[1-(adamantane-1-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
(2S,4R)-4-amino-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-N-methylpyrrolidine-2-carboxamide
ethyl 1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine-3-carboxylate
N-(3-methoxyphenyl)-3-[1-(pyridazine-4-carbonyl)piperidin-4-yl]propanamide
N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-[(dimethylamino)methyl]-1-{[4-(2-phenylethoxy)phenyl]methyl}azepan-4-ol
3-(3-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-4-methylpyridine
methyl 6-({cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-(furan-3-amido)thieno[2,3-b]pyridine-2-carboxylate
N-[3-(4-tert-butylphenoxy)-2-hydroxypropyl]-4-chloro-1-methyl-1H-pyrazole-5-carboxamide
N-(4-{[(4-methoxypyridin-2-yl)methyl](methyl)carbamoyl}phenyl)-2-methylfuran-3-carboxamide
[(3R,4R)-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(1S,6R)-9-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S,4R)-N-(4-acetylphenyl)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carboxamide
methyl({[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
2-[1-(3-methylpyridin-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
3-{[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4-propyl-4H-1,2,4-triazole
N-methyl-2-[(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]acetamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
2-[4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]pyrimidine
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
(1R,5R)-3-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(5-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}pyrimidin-2-yl)amino]acetic acid
N,N-dimethyl-2-[(3-phenylbutanamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(4S,4aS,8aS)-1-(furan-3-carbonyl)-4-phenyl-decahydroquinolin-4-ol
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
3-(4-benzyl-1H-pyrazol-5-yl)-1-(thian-4-yl)piperidine
4-{2-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
N-[(2S,4R,6S)-2-(2,4-dimethoxy-3-methylphenyl)-6-(2-methylpropyl)oxan-4-yl]acetamide
1-(2-aminoethyl)-N-[(1S,2R)-2-(hydroxymethyl)cyclopentyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-methylpyridin-4-yl)-4-[(2,3,6-trifluorophenyl)methyl]piperazine
N-[(2-fluorophenyl)methyl]-5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
N-[(4-hydroxyazepan-4-yl)methyl]-2,3-dimethyl-1H-indole-7-carboxamide
5-cyclobutanecarbonyl-1'-(5-fluoropyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{[4-(2-chlorophenyl)-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-methyl-N-[1-(3-methylphenyl)piperidin-4-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl})amine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-({3-methyl-7-[(2E)-4-methylpent-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
N-cyclohexyl-3-{[(2-cyclopropylphenyl)carbamoyl]amino}propanamide
N-ethyl-2-{[2-(1H-indol-1-yl)ethyl](methyl)amino}pyridine-3-carboxamide
3-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
3-[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]benzoic acid
N-cyclopentyl-4-[(oxan-3-yl)sulfamoyl]benzamide
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-6-methylphenol
N-methyl-1-(piperidin-3-ylmethyl)-N-(quinolin-8-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(benzyloxy)-1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
N-[3-(cyclohexylsulfanyl)propyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
2-methoxy-3-{[(piperidin-4-yl)amino]methyl}-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one