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1-(2-chlorophenyl)-4-[(2,4-dimethoxy-3-methylphenyl)methyl]piperazin-2-one
2-{4-[1-(4-methoxyphenyl)piperidin-4-yl]-1-methylpiperazin-2-yl}ethan-1-ol
1-(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-1,4-diazepan-1-yl)ethan-1-one
2-{1-[(3-methoxyphenyl)methyl]-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl}ethan-1-ol
3-[(3-chlorophenyl)methyl]-1-(6-ethylpyrimidin-4-yl)piperidine-3-carboxylic acid
4-(1H-imidazol-2-ylmethyl)-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
(3S,4R)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-3-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(4-ethenylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-{[4-(methylsulfanyl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
9-[2-hydroxy-3-(2-methylphenoxy)propanoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-6-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-benzoxazole
(1S,5R)-3-benzyl-6-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-cyclobutanecarbonyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine-4-carboxamide
3-methyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
2-[3-(2-methyl-1H-imidazol-1-yl)propanamido]-N-(pyridin-2-ylmethyl)benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-(4-methylpiperidin-1-yl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole-5-carboxamide
N-[1-(1-{[(1-methyl-1H-pyrazol-4-yl)carbamoyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)ethyl]acetamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1,8-naphthyridine-2-carboxamide
3-[(3-methoxypyrrolidin-1-yl)sulfonyl]-N-(2,2,2-trifluoroethyl)benzamide
N-(3-{4-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]piperidin-1-yl}phenyl)-4-phenylbutanamide
7-{4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinoxalin-2-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)butanamide
3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
N-[(3R)-1-benzylpyrrolidin-3-yl]-2-cyclopropyl-4-hydroxy-N-methylpyrimidine-5-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(furan-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-(2-{[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-(3-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(piperazin-1-yl)ethyl]amino}methyl)piperidin-2-one
4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)thiomorpholine
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
(2R)-2-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-methylbutan-1-one
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
ethyl 2-{1-[2-(pyridin-3-yl)acetyl]piperidin-2-yl}acetate
2-(4-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-amine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethyl-2-oxoimidazolidine-4-carboxamide
3-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
3-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}-1-[2-(pyridin-2-ylsulfanyl)ethyl]urea
1-[(2-aminopyridin-3-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(2R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(methoxymethyl)pyrrolidine
5-methoxy-N,3-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
2-cyclopropyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-(3-hydroxypropyl)-8-[(4-methoxy-2-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(3-phenylpropyl)benzamide