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N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(methylsulfanyl)propanamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})amine
(4aS,7aR)-1-[2-(1-ethylpiperidin-4-yl)acetyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(3-fluorophenoxymethyl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
N-[(3R,4S)-1-(2-amino-2-methylpropyl)-4-propylpyrrolidin-3-yl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-(2-{1-benzyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)pyrazine
7-(cyclobutylmethyl)-2-[2-(morpholin-4-yl)-2-oxoethyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(5-methoxyfuran-2-carbonyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
(2S,3S)-3-methyl-2-{[2-(propan-2-yl)pyrimidin-5-yl]formamido}pentanamide
N-(5-{[methyl(pyridin-3-ylmethyl)amino]methyl}pyrimidin-2-yl)benzenesulfonamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-(carbamoylmethyl)-N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}piperidine-4-carboxamide
(2R)-2-amino-N-{[(4-fluoro-2-methylphenyl)carbamoyl]methyl}-4-methylpentanamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(thiophen-2-ylmethyl)amino]benzamide
1-(1-{1-[(3-chloro-4-methoxyphenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
2-ethoxy-3-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
2-(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N,N-dimethyl-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-sulfonamide
8-(pyrimidin-2-ylmethyl)-8-azaspiro[4.5]decane-7,9-dione
(4aR,8aR)-2-(2,1,3-benzothiadiazol-5-ylmethyl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
1-(1-ethylpiperidin-4-yl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-ethyl-3-{2-[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
7-(cyclopropylmethyl)-2-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanoyl}-2,7-diazaspiro[4.5]decan-6-one
(4aS,8aR)-1-(3-aminopropyl)-6-[5-(methoxymethyl)furan-2-carbonyl]-decahydro-1,6-naphthyridin-2-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3-hydroxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[(4-fluorophenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
6-(azocane-1-carbonyl)-N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethylfuran-3-carboxamide
methyl 6-{[(2-methoxyethyl)(thiophen-2-ylmethyl)amino]methyl}pyridine-2-carboxylate
4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
(1R,5R)-3-(2,4-dimethylpyrimidine-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-hydroxybutyl)-5-methoxybenzamide
1-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-methyl-N-[2-(pyridin-2-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-benzoyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-(2-oxoazepan-3-yl)-3-propyl-1H-pyrazole-5-carboxamide
3-methoxy-1-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
N-methyl-3-propyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
methyl[(2E)-2-methylbut-2-en-1-yl]({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
ethyl 4-[(4-chlorophenyl)methyl]-1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine-4-carboxylate
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
N,5-dimethyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
2-(3-fluorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
2-{5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-pyrazol-3-yl}phenol
2-{5-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol