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9-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-{6-[benzyl(methyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperidin-3-yl)methyl]acetamide
N-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]piperidin-4-yl}methanesulfonamide
3-(1H-indazol-7-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)urea
2-[benzyl({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-methoxyphenol
3-[3-({[1-(methoxymethyl)cyclopentyl]carbamoyl}amino)phenyl]-N-methylpropanamide
N-({7-[(2-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
6-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-N-(1-methoxybutan-2-yl)-5-methylthieno[2,3-d]pyrimidin-4-amine
2-ethyl-5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
5-(2,6-difluorophenoxymethyl)-N-[1-(3-methoxyphenyl)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
N'-(3-ethylphenyl)-N-[(3,4,5-trimethoxyphenyl)methyl]butanediamide
2-[benzyl(methyl)amino]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
2-{2-[(2-methyl-3-oxopiperazin-1-yl)methyl]phenyl}-6-(2-phenylethyl)-3,4-dihydropyrimidin-4-one
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
3-(2-hydroxyphenyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
3-(1,3-benzothiazol-2-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]propanamide
N-methyl-N-[(3-methyloxetan-3-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
8-(furan-3-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]piperazine-2-carboxylic acid
N-cyclopropyl-4-(2,2-diphenylethyl)piperazine-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
2-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]acetamide
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-[2-(pyrrolidin-1-yl)ethyl]piperidine-4-carboxamide
5-cyclopropanecarbonyl-1'-[(2,3-difluoro-4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclopropyl-1-(1-ethylpiperidin-4-yl)piperidine-3-carboxamide
N-methyl-N-(quinolin-5-ylmethyl)-3,4-dihydro-2H-1-benzopyran-2-carboxamide
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
methyl 3-(3-methoxybenzamido)-5-[(pyridin-3-ylformamido)methyl]benzoate
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(pyridine-2-carbonyl)piperidine-2-carboxamide
1,9-dimethyl-4-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aS,7aR)-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[2-(4-chlorophenyl)morpholin-4-yl]-4-oxobutane-1-sulfonamide
N-{[(2S,4S)-1-[ethyl(methyl)sulfamoyl]-4-fluoropyrrolidin-2-yl]methyl}morpholine-4-carboxamide
1-(2-benzylphenyl)-3-[(1R,2S)-2-hydroxycyclohexyl]-3-methylurea
6-{[(thiophen-2-ylmethyl)amino]methyl}-1,4-oxazepan-6-ol
3-methyl-5-({4-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1,2-oxazole
5-ethyl-N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(2,3-dihydro-1H-inden-5-yl)-1-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}urea
3-{[({6,7-dimethoxy-2-[(4-methylphenyl)methoxy]quinolin-3-yl}methyl)amino]methyl}-1λ6-thiolane-1,1-dione
2-(5-ethyl-1,3-oxazole-4-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6-[4-(cyclopropylmethyl)piperazin-1-yl]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
5-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]carbamoyl}-1H-imidazole-4-carboxylic acid
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[4-(methylamino)piperidin-1-yl]methyl}piperidin-2-one
N-ethyl-2-(pyrazin-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
methyl 1-({3-[(2-oxo-2,3-dihydro-1H-indol-5-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxylate
1-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
1-[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
7-(2-methoxyphenyl)-2-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-3-(pyridin-3-yl)propanamide