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5-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
2-methyl-4-(2-methylphenyl)-1-[1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]piperazine
7-(3-chlorophenyl)-4-[2-(1H-imidazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-methoxyphenoxymethyl)-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(trifluoromethyl)benzene-1-sulfonamide
(2R)-2-hydroxy-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-phenylethan-1-one
2-[3,5-dimethyl-4-({methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
N-(1-benzylpiperidin-4-yl)-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
(3S,4S)-1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-ethyl-6-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
(1S,2S)-2-{4-[(3-ethyl-5-methyl-1,2-oxazol-4-yl)methyl]piperazin-1-yl}cyclohexan-1-ol
2-(2H-1,3-benzodioxol-5-yl)-1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]ethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-fluorophenyl)ethyl]acetamide
N-(furan-2-ylmethyl)-5-(methoxymethyl)-N-(3-methylbutan-2-yl)furan-2-carboxamide
9-methoxy-N-(3-methylbutyl)-7-oxo-3-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2E)-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-3-yl)prop-2-en-1-one
(1S,3R)-3-amino-N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]cyclopentane-1-carboxamide
2-(1-methyl-1H-indazol-3-yl)-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
4-(1H-pyrazol-1-yl)-1-[2-(thiophen-3-yl)acetyl]piperidine-4-carboxylic acid
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
1-ethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1H-indole-5-carboxamide
N-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-(furan-2-yl)pyrrolidine-1-carboxamide
N-(cyclopentylmethyl)-4-(3-hydroxy-3-methylbutyl)benzamide
3,5-dichloro-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-4-methylbenzamide
8-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
8-{[2-(trifluoromethoxy)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
5-(1-benzofuran-2-yl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2,4-triazin-3-amine
(1S,5R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]propan-1-one
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(oxan-4-yl)-1,4-diazepan-2-one
8-benzyl-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{4-[(2,5-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
3-[2-(1-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]benzonitrile
6-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]pyrazine-2-carboxamide
3-{2-oxo-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-(cyclohex-3-en-1-ylmethyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-[(2R,3R)-1'-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-[({4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}methyl)amino]ethan-1-ol
N,2-dimethyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(3-chloro-4-hydroxyphenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1-[1-(azepan-1-yl)-1-oxopropan-2-yl]-3-methoxy-1,2-dihydropyridin-2-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[2-(thiophen-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
3-{5-[2-(2,4-dioxoimidazolidin-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(propan-2-yl)propanamide
1-[cyclohexyl(methyl)amino]-3-(3-{[4-(dimethylamino)piperidin-1-yl]methyl}phenoxy)propan-2-ol