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2-{1-[(4-ethoxyphenyl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
1-methyl-2-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-(6-methoxyquinolin-8-yl)urea
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(oxolan-2-ylmethyl)piperazine
2-cyclopentyl-1-(3-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxymethyl}piperidin-1-yl)ethan-1-one
1-[1'-(3,5-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N5-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(4-{[1-(1-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
3-[5-(1H-imidazol-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
3-cyclohexyl-N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1H-pyrazole-4-carboxamide
1-{4-[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]urea
3-(hydroxymethyl)-1-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperidin-3-ol
3-({[(2-chloropyridin-3-yl)methyl](methyl)amino}methyl)-1-(cyclobutylmethyl)-3-hydroxypiperidin-2-one
3-(1H-imidazol-1-ylmethyl)-N-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carboxamide
2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}-N-(1,3-thiazol-2-yl)propanamide
1-cyclohexyl-N-[2-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
pyridin-3-yl(4-{[3-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
1-methyl-3-(piperidine-1-carbonyl)-N,N-bis(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methyl-6-[2-(pyridin-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
2-(4-acetylphenoxy)-N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
methyl 3-{1-benzyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}benzoate
2-(6-methoxypyridin-3-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
N-ethyl-15-methyl-N-(2-methylprop-2-en-1-yl)-13-oxo-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
4-(7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl)morpholine
(1R,5R)-6-[(3,4-dimethoxypyridin-2-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[2-(4-carboxypiperidin-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-(3-carbamoylpyridin-2-yl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
1-[2-(benzylsulfanyl)ethyl]-3-(1,3-dimethyl-1H-pyrazol-5-yl)urea
2-(1-cyclopropanecarbonylpiperidin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2S,4S)-4-amino-N,N-diethyl-1-[2-(1H-indazol-3-yl)acetyl]pyrrolidine-2-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-phenyl-1,3-thiazol-2-yl)piperidin-3-ol
2-(3-methoxypropyl)-9-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(1H-pyrazol-1-yl)ethyl]-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
propan-2-yl 3-{[2-(4-methoxyphenyl)phenyl]carbamoyl}piperidine-1-carboxylate
2-[5-(3,4-dihydro-2H-1-benzopyran-3-yl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
4-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}-2-ethoxyphenol
2-{2-methoxy-5-[(2-methyl-4-phenylpiperazin-1-yl)methyl]phenoxy}acetic acid
N-methyl-N-(piperidin-4-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(cyclohexylmethyl)-N-[(4-ethylphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
8-[2-(2,5-dimethylphenyl)acetyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)ethan-1-one
3-(2,5-dimethoxyphenyl)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidine
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one