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4-({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}amino)-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
3-{1-[(4-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1-[2-(piperidin-1-yl)ethyl]urea
1-[benzyl(methyl)amino]-3-[4-({[3-(propan-2-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
2-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)pyridine
5-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-3-(propan-2-yl)-1,2-oxazole
N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N,5,7-trimethyl-N-(propan-2-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
1-{4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperazin-1-yl}-2-phenoxyethan-1-one
1-[5-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-cycloheptyl-N-[2-(4-methylphenyl)propan-2-yl]-6-oxopiperidine-3-carboxamide
1-(4-phenyl-1,4-diazepan-1-yl)-4-(piperidin-1-yl)butan-1-one
2-chloro-N-ethyl-N-(propan-2-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
[(3,5-dichloropyridin-4-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
2-ethoxy-5-[2-(4-methoxyphenoxymethyl)pyrimidin-4-yl]benzoic acid
3-[(1-acetylpiperidin-4-yl)oxy]-N-(1-cyclopropylethyl)-4-methoxybenzamide
2-[(4-benzoylpiperazin-1-yl)methyl]quinolin-8-ol
5-benzyl-N-(1,4-dioxan-2-ylmethyl)-N-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-ethyl-1-methyl-3-{1-[2-(oxan-2-ylmethoxy)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl](pyridin-2-yl)methanol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-2-methoxypyridine-4-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(1,3-thiazol-2-ylmethyl)pyrimidin-2-amine
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N,5-dimethyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
(2S,4R)-4-amino-1-[(1,4-dimethylpiperidin-4-yl)methyl]-N-methylpyrrolidine-2-carboxamide
1-(3-phenylpropyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
4-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
[(1-cyclopentylpiperidin-3-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl][2-(piperidin-1-yl)ethyl]amine
2-(5-ethyl-1,3-oxazole-4-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
4'-(oxan-2-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 4-({4-[2-(4-fluorophenyl)acetyl]-7-oxo-1,4-diazepan-1-yl}methyl)benzoate
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
1-[(5-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}thiophen-3-yl)methyl]pyrrolidine
1-[4-(dimethylamino)azepan-1-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
13-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
[4-(5-phenyl-1,2-oxazole-3-carbonyl)-1,4-oxazepan-6-yl]methanol
2-{2-[2-(furan-3-yl)-1H-imidazol-1-yl]ethyl}-4,5-dimethyl-1H-1,3-benzodiazole
(1R,5R)-6-(cyclobutylmethyl)-3-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonane
3-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-1-methyl-1-[2-(4-methylphenoxy)ethyl]urea
3-(2-amino-1,3-thiazol-4-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-5-cyclopropyl-1H-pyrazole-3-carboxamide
1-(oxan-4-ylmethyl)-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
[2-(2-chlorophenoxy)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-[(3S,4R)-1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
6-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]pyrimidin-4-ol
ethyl 2-{2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}pyridine-3-carboxylate
5-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
N-{[6-(2-ethylphenyl)pyridin-3-yl]methyl}acetamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
4-[4-(oxolan-2-ylmethoxy)phenyl]-4H-1,2,4-triazole
N-[(5-fluoro-2-methylphenyl)methyl]-3-methoxy-2,2-dimethylpropanamide