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N-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]azocane-1-carboxamide
2-methyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-methoxypropan-1-one
methyl 5-[3-(1,2-oxazinan-2-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1R,5R)-6-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-[2-hydroxy-3-(piperazin-1-yl)propyl]-1H-1,2,3-triazole-5-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(2,3,6-trifluorobenzoyl)piperidin-3-yl]propanamide
[4-(3-phenoxybenzoyl)-1,4-oxazepan-6-yl]methanol
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
4-[(dimethylcarbamoyl)methyl]-N-(2-phenylphenyl)-1,4-diazepane-1-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-(naphthalen-2-ylmethyl)piperidine-4-carboxamide
ethyl 3-{2-[4-(2H-1,3-benzodioxole-5-amido)-1H-pyrazol-1-yl]acetamido}-5-methylhexanoate
1-methyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
2-[(4-chlorophenyl)methyl]-8-[(4-methyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N4-(1-cyclopropanecarbonylpiperidin-3-yl)-5,6-dimethylpyrimidine-2,4-diamine
(4S)-4-acetamido-5-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-5-oxopentanamide
2-(4-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrimidine
(1R,5S)-3-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3,4-dimethoxyphenyl)-1-(4-methylpyrimidin-2-yl)piperidin-3-amine
1-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
1-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,2,3,6-tetrahydropyridine
ethyl 5-(1-methoxypropan-2-yl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-N-(propan-2-yl)pyridine-4-carboxamide
4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-3,5-dimethylphenol
6-{2-[(dimethylamino)methyl]phenoxy}-N-ethyl-N-methylpyridine-3-carboxamide
2-{[5-(2H-1,3-benzodioxol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methyl-1,3,4-oxadiazole
1,3-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3S,4S)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(naphthalen-2-yl)piperidin-3-ol
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
5-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-4-methylpyrimidine
N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-3-(piperazine-1-sulfonyl)benzamide
2,2-dimethyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
[(3R,4R)-1-(4-methoxy-2-methylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-cyclopentyl-4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-4-oxobutanamide
(3S,9aR)-3-ethyl-8-(3-methylbutyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{5-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]-2-ethoxyphenyl}methanol
2-{[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzoic acid
3-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-methyl-N-(pyridin-2-ylmethyl)aniline
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
1-{4-[2-(3,4-dimethoxyphenyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
1-[1-(furan-3-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
2-[(4-methylphenyl)amino]-2-phenyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]propanamide
1-[(3S,4S)-3-(azocan-1-yl)-4-hydroxypyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
2-(3-phenylpropyl)-8-(3,3,3-trifluoropropanoyl)-2,8-diazaspiro[4.5]decan-3-one
4-propyl-5-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]pyrimidine
3-(pyrrolidine-1-carbonyl)-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]piperidine
4-(2-methoxyethyl)-3-{1-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
3-[cyclopentyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)carbamoyl]pyridin-1-ium-1-olate