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ethyl 2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
N-ethyl-N-[2-(3-methylphenoxy)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
methyl 5-cyano-2-methyl-6-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyridine-3-carboxylate
{[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}dimethylamine
1-(1H-imidazol-2-ylmethyl)-4-[(3-methylphenyl)methyl]piperazine
(1S,5R)-6-benzyl-3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(dimethylamino)ethyl]-2-methyl-N-[(2-methylphenyl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
6-{4-[3-(5-methylfuran-2-yl)butyl]piperazin-1-yl}-9H-purine
[(1-methyl-1H-imidazol-2-yl)methyl]({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})(propan-2-yl)amine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}acetamide
N-(propan-2-yl)-1-[(1s,4s)-4-(2-methyl-1,3-thiazole-4-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentyl-1,2-oxazole-3-carboxamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
1-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}piperidine
4-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-2-yl)methyl]morpholine
6-(3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropyl)-2,3,4,5-tetrahydropyridazin-3-one
(1R,5R)-3-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[1-(propan-2-yl)-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]pyridine
3-[1-(2-hydroxypyridin-3-yl)-1H-pyrazol-4-yl]propanoic acid
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N3-(4-fluorophenyl)-N5-[(4-methoxyphenyl)methyl]piperidine-3,5-dicarboxamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(trimethyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(5-{[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}thiophen-2-yl)acetamide
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
1-(4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenyl)-1H-pyrazole
2-(4-chloro-1H-indazol-1-yl)-N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)acetamide
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-3-methyl-1H-indole-2-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2,4-trimethylpyrimidine-5-carboxamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(3-methylpyridin-4-yl)methyl]acetamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-{6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}-4,6-dimethylpyridine-3-carbonitrile
(3aR,6aR)-2-methanesulfonyl-N-methyl-N-[2-(oxan-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(1-methyl-1H-indole-4-carbonyl)pyrrolidin-3-yl]methanol
4-(2-fluorophenoxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
(2E)-3-(3,5-difluorophenyl)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}prop-2-en-1-one
1-(2-{[(2-ethylpyrimidin-4-yl)methyl](methyl)amino}ethyl)piperidin-2-one
[(1-cyclohexylpiperidin-3-yl)methyl][(1-ethyl-1H-imidazol-2-yl)methyl](pyridin-3-ylmethyl)amine
9-(pyrimidin-2-ylmethyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2,4-dimethylphenoxy)-3-[2-(furan-2-yl)-1H-imidazol-1-yl]propan-2-ol
N-(butan-2-yl)-2-(pyrrolidin-1-ylmethyl)-N-(thiophen-3-ylmethyl)-1,3-thiazole-5-carboxamide
2-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-8-fluoroquinoline
1-[(3aR,6aR)-3a-[4-(4-acetylphenyl)piperazine-1-carbonyl]-octahydropyrrolo[3,4-c]pyrrol-2-yl]ethan-1-one
2-{1-[(3,4-difluorophenyl)methyl]-4-(1H-pyrazole-3-carbonyl)piperazin-2-yl}ethan-1-ol
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-1,4-diazepan-5-one
1-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 4-{[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
2,4-dimethoxy-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,3,5-triazine