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1-cycloheptyl-4-({[4-(2-hydroxyethoxy)phenyl]methyl}amino)pyrrolidin-2-one
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-benzyl{[2-(1H-imidazol-1-yl)pyridin-3-yl]amino}sulfonamide
N-(oxolan-2-ylmethyl)-3-{1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-4-yl}propanamide
3-(2-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-2-yl}ethyl)phenol
5-(pyrazin-2-yl)-1,2,3,4-tetrahydroisoquinoline
2-tert-butyl-6-(5-chloro-2-methoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N,N-dimethyl-1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}pyrrolidin-3-amine
(4aS,8aR)-6-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
4-(1-methyl-1H-pyrazol-4-yl)-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}pyrimidin-2-amine
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-2-methyl-1H-1,3-benzodiazole-5-carboxamide
6-cyclopropyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidin-4-amine
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3-propyl-1H-pyrazole-5-carboxamide
2-[(adamantan-1-ylmethyl)({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]ethan-1-ol
N-(1-cycloheptylpiperidin-3-yl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(2-methoxyphenyl)-5-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazole
(1-methoxypropan-2-yl)({[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl})amine
3-[(4-acetamidophenyl)methyl]-9-methoxy-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[1-(1-methyl-1H-indazol-5-yl)-1H-1,3-benzodiazol-2-yl]propanoic acid
5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
1-{4-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})(thiophen-3-ylmethyl)amine
4-[(4-fluorophenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoic acid
1-(4-acetylphenyl)-3-[2-(dimethylamino)ethyl]-3-[(5-methylthiophen-2-yl)methyl]urea
5-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
2-(6-chloro-2-fluoro-3-methoxyphenyl)-1H-imidazole
7-chloro-3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]quinolin-4-ol
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}piperidine-4-carbonitrile
(4aS,8aR)-1-butyl-6-(pyridine-3-sulfonyl)-decahydro-1,6-naphthyridin-2-one
2-[2-(pyridin-3-yl)ethyl]-9-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2,9-diazaspiro[5.5]undecan-3-one
(2R,3S,6R)-5-(1H-indazole-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{7-[(2,3-dimethoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}butane-1,2-dione
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methoxypiperidine
N-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
2-{[5-(4,5-dimethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methylpyrazine
7-methoxy-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-1,2,3,4-tetrahydronaphthalen-2-amine
(1R,5R)-6-benzyl-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
5-{methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}-1-[(2-methylphenyl)methyl]azepan-2-one
2-[3-oxo-2-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-butyl-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
2-(3-phenoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
2-[2-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[(2-phenoxyethyl)amino]methyl}phenoxy)propan-2-ol
(4aR,8aS)-6-(9H-fluoren-2-ylmethyl)-1-[(3-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one