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2-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amino}propan-1-ol
9-methyl-3-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-3,9-diazaspiro[5.6]dodecan-10-one
1-methyl-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
1-(4-methoxyphenyl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
N-(cyclopropylmethyl)-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-3-(pyrrolidine-1-carbonyl)piperazine
1-{7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecan-3-yl}-2-(dimethylamino)-2-(3-fluorophenyl)ethan-1-one
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]butanamide
2-[(3-{[2-(piperidin-1-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
2-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}azetidin-3-yl)pyridine
N-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
4-hydroxy-N-[3-(1H-indazol-1-yl)propyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
1-(2-oxo-2-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{1-[1-(benzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propanoic acid
N-[(2-aminopyrimidin-5-yl)methyl]-5-(2-chlorophenyl)-N-methylfuran-2-carboxamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
6-(2-fluorophenyl)-N-[2-hydroxy-2-(pyridin-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}propane-1,2-diol
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-(4-phenylbenzoyl)piperidine
2-{[2-(difluoromethoxy)phenyl]methyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
(4aR,8aR)-4-(7-fluoro-2-methylquinoline-4-carbonyl)-octahydro-2H-1,4-benzoxazine
2-(3-fluorophenyl)-2-{[3-(2-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}acetic acid
1-({5-[(4-methoxy-2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-phenoxypropanamide
N-[2-(furan-2-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-(5-phenyl-1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl]benzonitrile
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3,3,3-trifluoropropan-1-one
1-{[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
5-benzyl-4-(2-methoxyacetyl)-1-(3-methoxyphenyl)piperazin-2-one
1-(5-chloro-2-methoxyphenyl)-3-(propan-2-yl)-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazole
N-[2-(N-methylmethanesulfonamido)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
8-[(3-fluorophenyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-(2,2,2-trifluoro-1-phenylethoxy)ethan-1-one
N-[3-(4-fluorophenyl)propyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
8-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
(2S,4R)-4-amino-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2-{[2-(2-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-3-methoxyphenol
N,1-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-3-phenyl-1H-pyrazole-5-carboxamide
methyl (2S)-1-[9-methoxy-7-oxo-3-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
N-[3-(4-fluorophenyl)phenyl]-1-(thiophene-3-carbonyl)piperidine-3-carboxamide
(3S,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(2-oxo-8-{pyrazolo[1,5-a]pyridine-7-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-3-yl)propanoic acid
ethyl 4-(2-phenylethyl)-1-(3-phenylprop-2-yn-1-yl)piperidine-4-carboxylate
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-8-methoxyquinolin-2-amine