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1-{4-[(3R,4S)-3-[(6-methylpyrimidin-4-yl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]piperidin-1-yl}ethan-1-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}acetamide
1-tert-butyl-N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}pent-4-enamide
2,7-dimethyl-N-[1-(thian-4-yl)piperidin-4-yl]pyrazolo[1,5-a]pyrimidine-5-carboxamide
2-(3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(phenoxymethyl)-3,4-dihydropyrimidin-4-one
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
(2S,4R)-N-ethyl-4-[2-(4-hydroxyphenyl)acetamido]-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
3-{2-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-(1-benzyl-5-oxopyrrolidin-3-yl)-1-(2,4,6-trimethylpyridin-3-yl)urea
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
4-methyl-5-(prop-2-en-1-yl)-6-[4-(9H-purin-6-yl)piperazin-1-yl]pyrimidin-2-amine
2-[3-(dimethylamino)pyrrolidin-1-yl]-1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}ethan-1-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-5-fluoroquinazolin-4-amine
(3aS,6aS)-5-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[cyclohexyl(methyl)amino]-3-[3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
(4aS,7aR)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-methoxyphenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
2-amino-4-(4-hydroxy-3-methoxyphenyl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-{2-[4-(3,5-dimethylphenyl)-1H-1,2,3-triazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
6-({7-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-5,6-dihydro-1,6-naphthyridin-5-one
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(2-chloro-4,5-diethoxyphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
methyl 4-{[(5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-yl)amino]methyl}benzoate
{2-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]phenyl}methanol
1-{3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(3-methoxyphenyl)methyl]piperidin-3-yl)methanol
N-(1-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
(1r,4r)-4-{[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]amino}cyclohexan-1-ol
6-(aminomethyl)-2-methyl-N-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}pyrimidin-4-amine
2-methyl-4-[4-(propan-2-yl)piperazin-1-yl]-6-propylpyrimidine
3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)adamantan-1-ol
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(3-methylpyridin-4-yl)methyl]amine
4-{3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-(2-fluorophenyl)-7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-methylbutan-1-one
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-(furan-2-yl)-N-(oxolan-2-ylmethyl)prop-2-enamide
1-methyl-4-[(6-methylpyridin-2-yl)methyl]-2-phenylpiperazine
2-cyclopropanecarbonyl-8-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}pyrimidin-4-amine
(1R,4S)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
4-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1-(propan-2-yl)piperidine
2-(4-benzyl-2-methyl-3-oxopiperazine-1-carbonyl)-3,4-dihydroquinazolin-4-one
5-(4-cyclohexylphenyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2,4-triazin-3-amine
2-(4-{[4-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
(2Z)-2-fluoro-3-phenyl-1-[3-(phenylamino)piperidin-1-yl]prop-2-en-1-one
methyl 1-[(3R,5S)-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-methyl-N-[(3R,5S)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
[(4aS,8aR)-6-(5-methyl-1,3,4-oxadiazol-2-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol