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3-[1-(6-aminopyridine-2-carbonyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
2-cyclopropyl-8-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3-methoxyphenyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazole-5-carboxamide
2-[methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
N,2,7,8-tetramethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
3-{2-[(2-methylpropyl)(pyridin-2-ylmethyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[4-({4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}methyl)phenyl]acetamide
N-cyclopropyl-1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
4-(4-benzoylpiperazin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
2-[5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
(2E)-3-(3,4-dimethoxyphenyl)-1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-2-en-1-one
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
9-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-[2-(3-fluorophenyl)ethyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-hydroxy-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-methoxybenzamide
(1R,2S)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-propylcyclopropane-1-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
N-(4-methoxy-2-methylphenyl)-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)propanamide
2-(furan-2-yl)-N-[1-(pyridin-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(4-fluorophenyl)-4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1,4-diazepane
7-(4-phenyl-1,3-thiazole-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
methyl 5-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-{3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
1-(3,5-dimethylphenyl)-4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperazin-2-one
N,N-dimethyl-5-({3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)pyrimidin-2-amine
1-(4-phenyl-1H-imidazole-5-carbonyl)-2-(pyrrolidine-1-carbonyl)piperazine
methyl 1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]cyclopropane-1-carboxylate
2-ethyl-N-(2-methylbutyl)-2H-1,2,3,4-tetrazol-5-amine
2-(1-ethylpiperidin-4-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
4-ethyl-3-[(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
1-[(3R,4S)-3-[(2-amino-6-methylpyrimidin-4-yl)amino]-4-propylpyrrolidin-1-yl]-3-hydroxypropan-1-one
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(furan-3-ylmethyl)piperidine
(3S,4S)-1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
N-(2-{4-[(4-methyl-1H-imidazol-5-yl)methyl]morpholin-2-yl}ethyl)thiophene-3-carboxamide
[2-(2-methoxynaphthalen-1-yl)ethyl](1-methoxypropan-2-yl)amine
1-{6-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-3-yl}ethan-1-one
1-[benzyl(methyl)amino]-3-[5-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
6-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-ethyl-N-[(4-methoxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(1S,5R)-6-{[3-(methylsulfanyl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(cyclohex-1-en-1-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
N-{4-[4-(oxan-4-ylmethyl)-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepane-1-carbonyl]phenyl}acetamide
methyl 1-[(3R,5S)-1-[(4-methylphenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[(4aS,8aS)-decahydroisoquinoline-2-sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid