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4-(2-methoxy-3-methylbenzoyl)-2-(trifluoromethyl)morpholine
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(pyrazin-2-yl)piperazin-1-yl]propan-1-one
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2,5-dimethylphenyl)methyl]pyrimidin-2-amine
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-(2-ethylpyrimidin-5-yl)-6-methylquinoline
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(oxolane-2-carbonyl)piperazine
2-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)-6-methylquinolin-4-ol
2-[9-(5-cyano-4,6-dimethylpyridin-2-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
1-[(2,6-difluorophenyl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-cyclopentyl-2-(2-methyl-1H-imidazol-1-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)acetamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
4-ethyl-3-{1-[1-(pyrimidin-2-yl)piperidine-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
(4aS,8aR)-6-[2-amino-6-(methylamino)pyrimidin-4-yl]-1-propyl-decahydro-1,6-naphthyridin-2-one
3-{4-[1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]pyridin-2-yl}phenol
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(methylamino)pyridine-3-carboxamide
N-[(3S,4R)-1-(3-methoxybenzoyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl}ethan-1-ol
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-phenylpropan-1-one
2-(2-chloro-4-fluorophenoxymethyl)-4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,3-oxazole
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
1-methyl-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
methyl 2-[methyl(2-methylpropyl)sulfamoyl]-6-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1r,4r)-4-{[2-(dimethylamino)-2-(2-fluorophenyl)acetamido]methyl}cyclohexane-1-carboxamide
2-amino-6-(2-methoxyphenyl)-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-(cyclooctylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1S,5R)-6-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-(1-butyl-1H-imidazol-2-yl)-1-(1-methyl-1H-imidazole-2-carbonyl)piperidine
methyl 2-{[(4-methylphenyl)methyl]sulfamoyl}-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(2H-1,3-benzodioxol-5-yloxy)-1-(oxan-4-yl)piperidine-4-carboxylic acid
(2S,4S)-4-{4-[(3-cyclohexylpropanamido)methyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
1-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}cyclohexane-1-carboxamide
2-(dimethylamino)-N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-(3-methylphenyl)acetamide
N-[(2-fluorophenyl)methyl]-5-[(2-methoxyethyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-(pyridine-2-carbonyl)-1,4-diazepan-2-one
2-(4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(oxan-4-yl)piperazine
5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
7-(1-benzothiophen-3-yl)-4-(pyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(1H-1,3-benzodiazol-1-yl)-1-(6-cyanopyridin-2-yl)piperidine-4-carboxylic acid
5-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
3-[(2-fluorophenyl)formamido]-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
4-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(3-cyano-4-ethoxyphenyl)-3-(2-methanesulfonamidoethyl)urea
N-(3,4-difluorophenyl)-1-(3-methoxy-4-methylbenzoyl)piperidin-3-amine
N-[2-(3,5-difluorophenyl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-cyclopropyl-3-[1-(5-phenoxyfuran-2-carbonyl)piperidin-3-yl]propanamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine