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2-methyl-4-[4-(trifluoromethoxy)phenyl]-1H-imidazole
4-(1-methyl-1H-pyrazol-4-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidin-2-amine
2-[4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
5-acetyl-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-3-carboxamide
2-(4-methylphenyl)-5-(3-propylmorpholine-4-carbonyl)pyrimidin-4-ol
N-{[5-(2,1,3-benzothiadiazol-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
5-ethyl-6-methyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]thieno[2,3-d]pyrimidin-4-amine
5-methyl-N-[4-(5-methylfuran-2-amido)phenyl]pyridine-3-carboxamide
1-[2-({[2-(propylsulfanyl)pyrimidin-5-yl]methyl}amino)ethyl]piperidin-4-ol
5-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}pyrazin-2-ol
1-[4-(1H-pyrazol-4-yl)phenyl]piperazine
6-(4-methoxyphenyl)-N-(3-methoxypropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N'1-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}cyclopropane-1,1-dicarboxamide
5-{2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}pyrrolidin-2-one
2-{2-[1-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-(2-methylphenyl)-3-[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
2-(3-fluorophenyl)-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
2-{2-[1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
(3S,7S,8aS)-3-(4-aminobutyl)-7-{[(2,5-dimethylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-({1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}amino)butan-1-ol
4-cyclohexyl-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(6-methylpyridin-2-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-phenyl-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methoxyquinoline
(1S,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 4-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}thiophene-2-carboxylate
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]pyridin-3-amine
1-ethyl-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(cyclopropanesulfonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[1'-(oxan-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-(3-hydroxy-3-methylbutyl)-N-[(1r,4r)-4-hydroxycyclohexyl]benzamide
2-(ethylamino)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidine-5-carboxamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
N-(furan-3-ylmethyl)-N,5-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(1S,5R)-6-(3-methylbenzoyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(1-butyl-1H-imidazol-2-yl)-1-(4-chloro-2-fluorobenzoyl)piperidine
5-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)pyrimidine
N4-[(2-fluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
methyl 6-(4-phenylbutanoyl)-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methanesulfonyl-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-methyl-1-[1-(2-phenylethyl)azetidin-3-yl]piperidine
N-[(2R,3R)-2-ethoxy-1'-(1,3-thiazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(2S)-2-hydroxy-3-phenyl-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}[(5-methylfuran-2-yl)methyl]amine
2-{[4-(1-phenylethyl)-5-(1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
methyl 4-(3-acetamidophenyl)-3-methylbenzoate
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(pyridin-2-yl)acetamide