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2-[(2S,4S)-2-(diethylcarbamoyl)-4-(2-fluoro-4-methylbenzamido)pyrrolidin-1-yl]acetic acid
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopropyl-2-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}acetamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-methanesulfonamido-N-[(3R,4S)-4-propyl-1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]acetamide
(2E)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-3-phenylprop-2-en-1-one
N-[(4-fluorophenyl)methyl]-1-{2-[(2,3,4-trimethoxyphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-(2-methoxyethyl)-9-[3-(1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
6-fluoro-2-[(4-hydroxypiperidin-1-yl)methyl]quinolin-4-ol
4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}-1-phenylpiperazin-2-one
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-(2-methoxyethyl)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1-(2,4,6-trimethylphenyl)urea
N,N-diethyl-1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-amine
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
5-chloro-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]furan-2-carboxamide
2-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-2,3-dihydro-1H-indazol-3-one
(3aR,6aR)-2-(cyclohexylcarbamoyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-methoxypropyl)-6-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-cyclopentyl-4-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(1H-imidazol-1-yl)acetamide
4-[hydroxy(thiophen-2-yl)methyl]-N-[3-(4H-1,2,4-triazol-4-yl)phenyl]piperidine-1-carboxamide
2-(3-fluorophenyl)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
8-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-6-(1-benzofuran-2-ylmethyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}pent-4-enamide
(1R,3S)-7-(5-fluoro-4-methoxypyrimidin-2-yl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
N-cyclopropyl-2-(ethylamino)-N-[(2-methoxyphenyl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
N-(carbamoylmethyl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
3-{[(3-methyloxetan-3-yl)methyl]sulfamoyl}-N-(thiophen-2-ylmethyl)benzamide
4-(2H-1,3-benzodioxol-5-yl)-3-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoethyl}benzamide
N-{3-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]phenyl}pentanamide
2-ethyl-6-methyl-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
[1-(1-benzylpiperidin-4-yl)-2-(2-fluorophenyl)ethyl][(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-5,6,7,8-tetrahydroquinoxaline
(2S,4S)-4-amino-1-[4-(methylamino)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
8-(2,1,3-benzoxadiazol-4-ylmethyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}quinolin-8-ol
9-ethyl-1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 6-methyl-2-(2-methyl-5-oxo-1,4-diazepan-1-yl)pyrimidine-4-carboxylate
7-(4-fluorophenyl)-2-[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-{3-[2-(1-phenylethyl)-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
1-{5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
N1,N1-dimethyl-N4-[1-(3-phenylpropyl)piperidin-3-yl]piperidine-1,4-dicarboxamide
6-cyclopentyl-2-[4-({ethyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
2-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one