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N-ethyl-N-[(4-methoxyphenyl)methyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(5-methyl-1,3-benzoxazol-2-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-5-phenoxyfuran-2-carboxamide
N-(2-phenoxyphenyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carboxamide
2-(carbamoylamino)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
5-[1-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)pyrrolidin-2-yl]-N-methylthiophene-2-carboxamide
4-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-sulfamoylbenzamide
2-[(2S)-2-({6-methylimidazo[1,2-a]pyridin-2-yl}formamido)-3-phenylpropanamido]acetic acid
[(3aS,6aS)-2-[4-(trifluoromethyl)pyrimidin-2-yl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(furan-3-ylmethyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-(1-{[methyl(oxolan-3-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}propanamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-propyl-1,2-oxazole-4-carboxamide
5-(naphthalen-1-yl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1,2,4-triazin-3-amine
4-methoxy-N-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-6-ethoxy-1,2-dihydroquinolin-2-one
(1S,5R)-3-methyl-6-[4-(morpholine-4-carbonyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-{2,7-diazaspiro[4.5]decan-7-yl}-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(4-{[3-(pyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)-1H-1,2,4-triazole
N-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
ethyl 4-[4-(4-{[2-(morpholin-4-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
(3R,4R)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-ethylpiperidine-3,4-diol
(3S,4S)-1-{[3-(morpholin-4-yl)phenyl]methyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
7-methyl-2-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-cyclohexanecarbonylpiperidine
3-{[2-(3-methoxypropyl)piperidin-1-yl]sulfonyl}benzonitrile
(3S,4R)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
7-(1-benzothiophen-3-yl)-4-(3-fluorobenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S,9aR)-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl({4-[(1-methyl-1H-indol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)[2-(pyridin-2-yl)ethyl]amine
3-({[(4,6-dimethylpyridin-3-yl)methyl]carbamoyl}amino)-N-(2-methoxyethyl)-2-methylbenzamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-tert-butylacetamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
(3aS,6aS)-2-(oxan-4-yl)-5-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-(propan-2-yl)piperidine-1-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
(3R,4R)-1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-(3-benzoylpiperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-[3-(trifluoromethyl)phenyl]acetamide
3-{4-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propyl]piperazin-1-yl}-2,5-dimethylpyrazine
5-methoxy-1-methyl-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(2-methoxyphenyl)methyl]propylamine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)morpholine-4-carboxamide
6,8-dimethyl-2-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}quinolin-4-ol