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N-(2-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}quinolin-6-yl)acetamide
(1S,4S)-5-cyclobutanecarbonyl-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(4-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}piperazin-1-yl)-N-(propan-2-yl)acetamide
1-(3-chlorophenyl)-4-(1-ethyl-1H-indole-5-carbonyl)piperazin-2-one
ethyl[2-(1H-pyrazol-1-yl)ethyl]{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
6-{[(9H-fluoren-9-yl)amino]methyl}-1,4-oxazepan-6-ol
1-ethyl-4-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
(3aS,6aS)-2-cyclopropanecarbonyl-5-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
6-{4-[4-(propan-2-yl)piperazin-1-yl]phenyl}-3,4-dihydroquinazolin-4-one
7-[(4-fluorophenyl)methyl]-2-(propane-1-sulfonyl)-2,7-diazaspiro[4.5]decane
1-[(2-chlorophenyl)methyl]-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(4-fluorophenyl)-2-hydroxy-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
4-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-3-methyl-1-propyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3-benzyl-1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
N-[2-(2-methoxyphenyl)ethyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
(1s,4s)-4-{4-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
(2S,4R)-N-ethyl-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
4,4,4-trifluoro-1-(3-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)butan-1-one
N-(3,4-difluorophenyl)-1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-3-amine
2-{4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-1,3-benzoxazole
2-methanesulfonyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)acetamide
2-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
4-(1-benzofuran-2-carbonyl)-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(5-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-2-ethoxyphenyl)methanol
N3-(1-benzylpyrrolidin-3-yl)-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
(2R,6S)-4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
3-{2-[cyclopentyl(methyl)amino]ethyl}-1-(3-fluoro-4-methylphenyl)-3-methylurea
4-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
4-{1-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}pyridine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-cyclopentyl-4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
(2R,6S)-2,6-dimethyl-4-(5-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)morpholine
3-{[5-(2-methyl-1,3-thiazol-4-yl)-1,2-oxazol-3-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-diethylacetamide
2-benzyl-8-{[5-(hydroxymethyl)furan-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-methoxyethan-1-one
6-ethyl-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-2-methylquinoline-4-carboxamide
2-cyclopropanecarbonyl-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[2-(pyridin-2-yl)ethyl]-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]piperidin-2-one
1'-(1-methyl-1H-pyrazole-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(2-chloro-4-methoxyphenoxymethyl)-N-cyclobutyl-1H-pyrazole-3-carboxamide
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(6-methylquinolin-5-yl)pyridine-3-carbonitrile
2-methoxy-5-[5-(piperidine-1-carbonyl)furan-2-yl]pyridine
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(4-methoxypyrimidin-2-yl)pyrrolidin-3-yl]methanol
5-benzyl-5-(piperidin-4-yl)-3-(pyridin-4-ylmethyl)imidazolidine-2,4-dione
4-ethyl-3-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-({3-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol