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N-(1,3-thiazol-2-yl)-3-{[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]amino}propanamide
3-{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}benzoic acid
2-{5-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3S)-3-(dimethylamino)azepan-1-yl]ethan-1-one
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-(2,2,2-trifluoroethyl)piperidin-4-amine
2-(6-chloro-2-fluoro-3-methylphenyl)-1-(oxan-4-yl)-1H-imidazole
(4aS,8aR)-1-propyl-6-(quinoline-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)benzamide
(dicyclopropylmethyl)(methyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
methyl 3-(5-methylpyrazine-2-carbonyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[2-methyl-4-({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-methoxy-N-({7-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
8-chloro-2-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}amino)methyl]quinolin-4-ol
1-[2-(5-benzyl-4-phenyl-1H-imidazol-1-yl)ethyl]pyrrolidin-2-one
3-(hydroxymethyl)-1-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)piperidin-3-ol
[(5-ethylfuran-2-yl)methyl](methyl)[(2-methylpyridin-4-yl)methyl]amine
dimethyl(2-{[(1-methyl-1H-imidazol-2-yl)methyl][(2-methylphenyl)methyl]amino}ethyl)amine
2-(1H-imidazol-2-yl)-N-(thiolan-3-yl)benzamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[3-(2-methoxyphenyl)propanoyl]piperidine-4-carboxylate
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)acetamide
4-methyl-6-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)pyrimidin-2-amine
2-(2-aminoethyl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}quinazolin-4-amine
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,7-dimethyl-1H-indole-2-carboxamide
N-(2-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-[(3R,4S)-1-(3-fluoro-4-methylbenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}cyclopropane-1-carbonitrile
2-methoxy-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenol
1-[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]piperidin-3-ol
2-[5-(3-acetylphenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
(2H-1,3-benzodioxol-5-ylmethyl)({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})(pyridin-3-ylmethyl)amine
(2S,4S,5R)-5-(3-chlorophenyl)-4-{[2-(dimethylamino)ethyl]carbamoyl}-1-methylpyrrolidine-2-carboxylic acid
4-[3-(benzyloxy)azetidine-1-carbonyl]-1-ethylpyrrolidin-2-one
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-3-(2-methoxyphenyl)propanamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2,2,6,6-tetramethylpiperidin-4-amine
5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-{4-[(3-methylphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-[(1S,2R)-2-(cyclooctylamino)cyclobutyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
9-(2,4-dimethylquinoline-7-carbonyl)-3-oxa-9-azaspiro[5.5]undecane
1-butyl-3-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1-(pyridin-4-ylmethyl)urea
1-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,N-dimethyl-2-[(1S,5R)-3-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
ethyl (2S)-2-[2-(2,4-dimethylbenzenesulfonamido)acetamido]propanoate