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6-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-cycloheptyl-6-oxopiperidine-3-carboxamide
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(pyrrolidin-1-yl)piperidine
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-1-ethyl-6-oxopiperidine-3-carboxamide
4-({4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)benzoic acid
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2,6,8-trimethyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
1-(3-chlorophenyl)-4-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine
N,N,3-trimethyl-4-({[1-(6-methylpyridin-3-yl)ethyl]carbamoyl}amino)benzamide
N-cyclohexyl-N-methyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-phenyl-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
4-{4-[2-(3-fluorophenyl)acetyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
4'-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}pyridine
4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazine-1-sulfonamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(oxane-4-carbonyl)piperidin-3-yl]piperazine
1-[1-(propan-2-yl)piperidine-4-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
N-benzyl-3-{[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-4-[4-(3-methoxyphenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-methyl-6-(methylsulfanyl)quinoline
[7-chloro-5-(quinolin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-[5-(3-hydroxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-methyl-N-(propan-2-yl)piperidine-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzamide
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(thiophen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})amine
2-({[(8-methoxy-2H-chromen-3-yl)methyl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
4-(4-ethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-yl)morpholine
2-methanesulfonyl-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
methyl 2-(1-{7-acetamido-1-[(4-fluorophenyl)methyl]-1H-1,3-benzodiazole-5-carbonyl}-3-oxopiperazin-2-yl)acetate
8-(dimethyl-1,2-oxazole-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
5-{[2-(thiophen-2-yl)-1H-imidazol-1-yl]methyl}-2,1,3-benzothiadiazole
(1s,4s)-4-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}cyclohexan-1-ol
4-({3-[5-(piperidine-1-carbonyl)furan-2-yl]phenyl}methyl)morpholine
5-ethyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
6-cyano-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
ethyl 4-[3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanoyl]piperazine-1-carboxylate
4-[(1-{[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]morpholine
3-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
(3S,9aR)-8-[(3,4-dimethylphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-tert-butyl-6-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]-1,2-dihydropyrimidin-2-one
5-{1-[2-(piperidin-1-yl)acetyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-{2-[2-(2-methoxyphenyl)acetamido]ethyl}-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
ethyl 4-{2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetyl}piperazine-1-carboxylate
4-methoxy-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide