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N-ethyl-6-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{[(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)carbamoyl]amino}-N-methyl-2-phenylacetamide
3-(2-methoxyphenyl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
2-{4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
3-benzyl-4-[4-(4-chlorophenyl)butanoyl]piperazin-2-one
1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-4-(pyrrolidin-1-yl)piperidine
7-(8-methylquinolin-5-yl)-1,2-dihydroisoquinolin-1-one
N-benzyl-5,6-dimethyl-N-[(1R,3S,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidin-2-one
N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
1-benzyl-4-(2-cyclohexylethyl)-1,4-diazepan-6-ol
2-methoxy-6-[2-(pyridin-2-yl)ethyl]-3-{[(thiolan-3-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
2,5-dimethoxy-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzene-1-sulfonamide
N-(1-methyl-1H-pyrazol-3-yl)-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}acetamide
2-[3-(2-methylpyrimidin-4-yl)phenoxy]propanamide
1-[2-({2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl}formamido)ethyl]piperidine-3-carboxamide
N-[1-(4-methanesulfonylphenyl)ethyl]-2-(methylamino)pyrimidine-5-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-2-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine
N-({3-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]furan-2-carboxamide
1-[1-({2-oxo-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-8-yl}methyl)piperidin-4-yl]pyrrolidin-2-one
4-[2-(2-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
methyl 3-(2-chlorobenzenesulfonamido)-5-{[2-(3-fluorophenyl)acetamido]methyl}benzoate
2-({2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenyl}amino)acetic acid
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-[5-(4-methylphenyl)furan-2-yl]propan-1-one
4-(2,5-dimethoxybenzoyl)-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
methyl (2S,4S,5R)-1,2-dimethyl-4-{[(5-methyl-1,2-oxazol-3-yl)methyl]carbamoyl}-5-(2-methylphenyl)pyrrolidine-2-carboxylate
1-[(3-fluorophenyl)methyl]-3-{[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
ethyl 3-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}carbamoyl)amino]propanoate
6-[6-hydroxy-4-(thiophene-2-carbonyl)-1,4-diazepan-1-yl]pyridine-3-carboxamide
5-methoxy-2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-methyl-1H-indole
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-4-hydroxy-3-methoxybenzamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
2-(4-fluorophenyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-methyl-9-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{[5-(1,2-dihydroacenaphthylen-5-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
7-(2-hydroxyethyl)-2-[(5-phenylthiophen-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
9-methoxy-7-oxo-3-[2-(propan-2-yl)oxane-4-carbonyl]-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(2-methoxyphenyl)pyridazine
3-(azepane-1-carbonyl)-1-ethyl-N-methyl-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-hydroxy-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(4-methylphenyl)pyrimidine-5-carboxamide
1-(cyclohexylmethyl)-4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
(4aS,7aR)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-methylpyridin-4-yl)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,4-diazepane
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxyacetamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
7-(2,2-diphenylethyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine