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8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(2-methoxyphenoxy)piperidine
4-(8-fluoro-4-oxo-1,4-dihydroquinoline-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-(2-ethoxyphenyl)-3-oxo-3-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]propanamide
ethyl 2-[1-(1-benzofuran-3-carbonyl)piperidin-2-yl]acetate
N-methyl-N-[2-(pyridin-2-yl)ethyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-(3,4-dimethylphenyl)-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]-2-fluorobenzonitrile
(2E)-3-(3-fluorophenyl)-N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}prop-2-enamide
2-[3-phenyl-5-(pyridin-2-ylmethyl)-1H-1,2,4-triazol-1-yl]pyridine
2-amino-6-(1H-indol-3-yl)-4-[2-(2-methoxyethyl)pyrimidin-5-yl]pyridine-3-carbonitrile
(1R,5R)-3-(pyrazine-2-carbonyl)-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]-N-[(3,4,5-trimethoxyphenyl)methyl]propanamide
(2S,4S)-4-amino-N-methyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]pyrrolidine-2-carboxamide
2-methyl-4-{4-[2-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-(3-hydroxypropyl)-8-(quinolin-6-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(2H-1,3-benzodioxol-5-yl)-3-(4-methyl-1H-imidazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(dimethylamino)pyrimidin-2-yl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3aS,6aR)-3-[2-(piperidin-1-yl)ethyl]-5-(pyrimidin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-({2,5-dimethyl-3-[(2-methylpiperidin-1-yl)methyl]phenyl}methyl)-4-methyl-1,4-diazepan-5-one
4-[(prop-2-en-1-yl)sulfamoyl]-N-(quinoxalin-6-yl)benzamide
N,N-dimethyl-1-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-3-amine
2-{4-[(4-methylpiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
8-methyl-2-propyl-N-[2-(pyrazin-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N,N-dimethyl-1-({4-[2-(morpholin-4-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}methyl)cyclopentan-1-amine
N-(2-ethoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1-methyl-5-(thiophen-2-yl)-1H-pyrazole
4-[5-(propan-2-yl)pyrimidin-4-yl]piperazine-2-carboxylic acid
N-tert-butyl-2-[4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)phenoxy]acetamide
N-(2-ethoxyethyl)-3-{[(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}benzamide
1-[(4-fluoro-3-methoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-[2-(methylsulfanyl)phenyl]-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-3-ylmethyl)urea
N-(1,3-benzoxazol-2-ylmethyl)-4-methyl-1H-imidazole-2-carboxamide
N1-[4-(1H-imidazol-1-yl)phenyl]-N2-methylpyrrolidine-1,2-dicarboxamide
3-hydroxy-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]acetamide
(1R,5R)-3-methanesulfonyl-6-(5-phenyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)morpholine-4-carboxamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
1-benzyl-4-{[6-(dimethylamino)pyridin-3-yl]methyl}-1,4-diazepan-6-ol
N,2-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{9-[(4-ethylphenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
6-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]pyridine-2-carbonitrile
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(pyrrolidine-1-carbonyl)pyrazine
methyl 5-[(1-acetylpiperidin-4-yl)amino]-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate