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1-(4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-3-methylphenyl)-1H-pyrazole
3-(2-fluorophenyl)-6-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(1-cycloheptylpiperidin-3-yl)-5-cyclopropyl-1,3-oxazole-4-carboxamide
2-[1-(2-methylpropyl)-4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-2-yl]ethan-1-ol
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-1,7-dimethyl-1H-indole-2-carboxamide
4-{1-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-[3-(4-fluorophenyl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidine-2-carboxamide
2-(1'-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl)acetamide
(4aS,8aR)-1-(2-methylpropyl)-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-2-one
(2S)-2-({[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amino)propanamide
4-(benzyloxy)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
3-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}-4H-chromen-4-one
methyl 4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}benzoate
1-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyridin-2-amine
3-(5-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-N-(2-hydroxyethyl)propanamide
7-chloro-3-(morpholin-4-ylmethyl)-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
2-(3-{[methyl({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})amino]methyl}piperidin-1-yl)ethan-1-ol
2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrazine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
2-acetyl-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(cyclopropylmethyl)acetamide
5-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
6-(3-fluorophenyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-oxo-1-(prop-2-en-1-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrrolidine-3-carboxamide
(1S,5R)-3-(3-chlorobenzenesulfonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-(4-cyclopentylpiperazin-1-yl)-3-(2-hydroxyphenyl)-3-(4-hydroxyphenyl)propan-1-one
4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]pyrimidine-5-carboxamide
1-ethyl-5-methyl-N-[3-(3-oxopiperazin-1-yl)propyl]-1H-pyrazole-4-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-acetamidobenzamide
2-hydroxy-4-(methylsulfanyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}butanamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-[(3-methylphenyl)methyl]-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
5-(3-fluorophenoxymethyl)-N-(2-hydroxyethyl)-N-propyl-1H-pyrazole-3-carboxamide
4-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-2,1,3-benzoxadiazole
N-methyl-N-[(5-methylfuran-2-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-(2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-oxoethyl)-5-methyl-2,3-dihydro-1H-indol-2-one
(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)-N-(6-methoxypyridin-3-yl)pyrrolidine-1-carboxamide
[2-(4-methoxyphenyl)ethyl]({[2-(2-methylphenyl)pyrimidin-5-yl]methyl})[(1-methylpiperidin-4-yl)methyl]amine
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]pyrimidin-4-amine
6-[4-(4-methylphenyl)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
(2-ethoxy-5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenyl)methanol
3-[2-(2-methylphenyl)ethyl]-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
3-(azepane-1-carbonyl)-N-cyclopropyl-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(3-methoxypropyl)-1-(4,4,4-trifluorobutanoyl)piperidine-3-carboxylic acid
(2-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide