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5-chloro-6-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyridine-3-carboxylic acid
2-(4-{[(3-propyl-1,2-oxazol-5-yl)methyl]amino}piperidin-1-yl)pyridine-4-carbonitrile
3-methyl-8-[1-(piperidin-4-yl)pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(furan-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]azepane
2-cyclopropyl-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-methylpyrimidine-5-carboxamide
1-(1-benzothiophen-2-ylmethyl)-3-(hydroxymethyl)pyrrolidin-3-ol
1-{5-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-[(2S)-2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-[(1S,5R)-3-[2-(4-fluorophenyl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-ethyl-9-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-ethyl-1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperidine-3-carboxylic acid
3-{2-amino-4-[4-(4-fluorophenoxy)piperidin-1-yl]-6-methylpyrimidin-5-yl}propanoic acid
1-(2-{1-[(3-chloro-2,6-difluorophenyl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
4-(furan-2-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{4-[6-(azepan-1-yl)pyridazin-3-yl]phenyl}ethan-1-one
7-(2-methylphenyl)-4-[(3-methylthiophen-2-yl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
6-methyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
2-tert-butyl-6-(2,3-dihydro-1-benzofuran-7-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-(carbamoylmethyl)-N-[1-(3,5-dichlorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
2-cyclopropyl-N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(1S,6R)-9-(isoquinoline-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
6-(cyclopent-1-ene-1-carbonyl)-1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octane
1-(1H-indol-2-ylmethyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
7-chloro-N,2-dimethyl-N-[2-(methylsulfanyl)ethyl]quinoline-4-carboxamide
ethyl 2-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-2-yl}acetate
2-(2,4-dichlorophenoxy)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]acetamide
1-(4-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonane-7-carbonyl}phenyl)imidazolidine-2,4-dione
2,3-dimethoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
(3R,5S)-5-[4-(benzenesulfonyl)piperazine-1-carbonyl]pyrrolidin-3-amine
(1R,5R)-6-(cyclopropylmethyl)-3-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-3,6-diazabicyclo[3.2.2]nonane
methyl 1-ethyl-5-{[1-(2-methoxyphenyl)propan-2-yl]amino}-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]pyridine-2-carboxylic acid
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(4-methoxyphenyl)-4-oxobutanamide
(1R,2R,6S,7S)-4-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(4aS,8aR)-6-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-ol
4-methyl-2-[4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
1-[2-({[(3-methyloxetan-3-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
(1S,5R)-6-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
8-chloro-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-2-carboxamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}ethan-1-one
2-[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-3-carboxamide
9-cyclopentanecarbonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1H-1,3-benzodiazol-2-ylmethyl)(methyl){[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
3-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-(2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(methylcarbamoyl)pyridin-2-yl]-4-phenoxypiperidine-4-carboxylic acid
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-3-[6-(methoxymethyl)pyridine-2-carbonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[({5-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol