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N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
N-cyclohexyl-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(2-chloro-6-methylphenyl)-2-methyl-2,8-diazaspiro[4.5]decane-8-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-(2-oxopiperidin-3-yl)pyrimidine-5-carboxamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-[4-(piperidin-1-ylmethyl)benzoyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-[2-(dimethylamino)pentyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[6-hydroxy-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-1-yl]methyl}benzoic acid
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(pyridin-3-ylformamido)ethyl]propanamide
2-{4-[4-(1H-pyrazol-1-yl)benzenesulfonyl]morpholin-3-yl}acetic acid
N4-(thiophen-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)isoquinoline
1-ethyl-3-(oxan-4-yl)-5-(5-phenoxyfuran-2-yl)-1H-1,2,4-triazole
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(indolizin-2-yl)pyridine-3-carbonitrile
N-[1-(cyclohexylmethyl)piperidin-3-yl]pyrazine-2-carboxamide
(4-{[5-chloro-2-(prop-2-en-1-yloxy)phenyl]methyl}morpholin-2-yl)methanamine
5-chloro-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
8-(3-methyl-1,2-oxazole-5-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4S)-1-[(6-methoxypyridin-3-yl)methyl]-4-methylpiperidine-3,4-diol
N-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
4-(1-hydroxypropyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
3-(3-methylpyridin-4-yl)quinoline
3-{[2-(hydroxymethyl)piperidin-1-yl]sulfonyl}-N-methyl-N-[2-(methylsulfanyl)ethyl]benzamide
N,5-dimethyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-cyclopropyl-8-[(4-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3S,4S)-4-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-1-(oxan-4-yl)pyrrolidin-3-ol
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[5-cyclopropyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(3-methoxyphenyl)pyrimidine
2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide
N-[4-(oxolan-2-ylmethoxy)phenyl]-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
4-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1λ6-thiomorpholine-1,1-dione
ethyl 1-[(2-methyl-1H-imidazol-4-yl)methyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
1-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
3-methoxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-(cyclohex-1-en-1-ylmethyl)-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}urea
(4aS,7aR)-1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(2-methylprop-2-en-1-yl)oxy]-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1,2,3,4-tetrahydroquinolin-2-one
2-[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-5-methoxy-1-methyl-1H-indole
2-[(3-hydroxypiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-phenyl-N-{1-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
6-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
ethyl 4-{6-[(5-chloro-2-hydroxyphenyl)methyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
1-ethyl-3-methyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
N-(5-acetamido-2-methylphenyl)-2-(2-hydroxyethyl)pyrrolidine-1-carboxamide
N-[2-(dimethylamino)ethyl]-4-methoxy-3-({1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}oxy)benzamide
4-(3-{[1-(1,3-thiazol-2-yl)piperidin-4-yl]oxy}benzoyl)morpholine