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N-(2-methoxyethyl)-1-methyl-N-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidin-4-amine
2-fluoro-5-sulfamoyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)benzamide
3-[methyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
1-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]ethan-1-one
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
2-(1H-imidazol-2-yl)-N-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide
2-[4-chloro-3-(trifluoromethyl)phenyl]-3-(pyrrolidine-1-carbonyl)pyridine
1-cyclopentyl-4-({2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)piperazin-2-one
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-methoxy-4-methyl-1,3-thiazole-5-carboxamide
2-(3-fluoro-4-methoxyphenyl)-2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]acetic acid
4-(1,4-dithiepan-6-yl)-2-[(3-methoxyphenyl)methyl]morpholine
1-(1-methylpiperidine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-(2-methylphenyl)-4-(2-methylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-({[(propan-2-yl)carbamoyl]methyl}sulfamoyl)-N-[(2R)-pyrrolidin-2-ylmethyl]benzamide
9-[2-(4-fluorophenyl)-2-hydroxyacetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[4-(6-methoxyquinolin-3-yl)-1H-pyrazol-1-yl]acetamide
methyl (2S)-1-{2-[4-(4-{[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
6-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}pyrimidin-4-amine
2-(methylsulfanyl)-1-[3-(4-phenylbenzoyl)piperidin-1-yl]ethan-1-one
ethyl 4-[1-(cyclohexylmethyl)-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-amido]piperidine-1-carboxylate
2-(1-methyl-1H-imidazol-2-yl)-1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazole
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(4-chlorophenyl)cyclobutane-1-carboxamide
N-[(1R,2S)-2-phenylcyclohexyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
(2S)-2-{[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-methylbutanamide
3-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
6-amino-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]hexan-1-one
2-(3-methyl-1H-pyrazol-1-yl)-1-[3-(2-phenylethyl)piperidin-1-yl]ethan-1-one
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-2,5-dimethylfuran-3-carboxamide
9-(cyclohex-3-en-1-ylmethyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[1-(pyridin-2-yl)ethyl]acetamide
3-cyclohexyl-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
4-methoxy-N-{1-[1-(oxan-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(2R,3R)-1'-(pyridin-2-yl)-3-(thiomorpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(3-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}phenoxy)acetamide
2-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]acetic acid
2-[4-(3-hydroxy-3-phenylpyrrolidin-1-yl)piperidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]propanamide
4-(1-acetylpiperidin-4-yl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
N-[(2R,4R,6S)-2-cyclohexyl-6-{3-methylimidazo[1,5-a]pyridin-1-yl}oxan-4-yl]acetamide
8-(3-chloro-5-fluoro-4-methoxyphenyl)-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]ethan-1-one
N,N-dimethyl-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrrolidin-3-amine
5-(2,3-dihydro-1H-isoindol-2-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
[(1-methyl-1H-imidazol-2-yl)methyl][(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
[2-methoxy-5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
3-(3-{3-[6-(dimethylamino)pyridazin-3-yl]phenyl}-1H-pyrazol-1-yl)propan-1-ol
ethyl 1-(2-methoxyacetyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
3-benzyl-4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperazin-2-one