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7-(2-hydroxyethyl)-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
N'-(2-fluoro-5-methylphenyl)-N-(2-methoxybutyl)butanediamide
1-(2,6-dimethylpyrimidine-4-carbonyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
1-[1-(3-methylbut-2-enoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
(3aR,5S,6S,7aS)-2-(1,3-thiazol-2-ylmethyl)-octahydro-1H-isoindole-5,6-diol
6-methyl-2-({methyl[4-(morpholin-4-yl)butyl]amino}methyl)quinolin-4-ol
1-[4-(2-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
(3S,4S)-4-methyl-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidine-3,4-diol
2-(4-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-2-oxopiperazin-1-yl)benzonitrile
1-tert-butyl-N-[3-(1H-indol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
5-phenyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
4-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}butanamide
N-[4-(6-methoxypyridin-3-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]cyclopentanecarboxamide
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)(quinoxalin-5-ylmethyl)amine
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]quinoxaline
2-methyl-N-[2-(5-methylfuran-2-yl)ethyl]imidazo[1,2-a]pyrimidine-3-carboxamide
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2,6-dimethylquinoline
1-(cyclohexylmethyl)-N3-ethyl-N5-[(1R)-1-(4-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-N-(2-methoxyethyl)thiophene-2-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(4-ethoxyphenyl)methyl](pyridin-3-ylmethyl)amine
N-methyl-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-N-(oxan-4-yl)acetamide
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-(6-methylpyridazin-3-yl)benzamide
2-chloro-5-fluoro-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzamide
1-(carbamoylmethyl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]piperidine-4-carboxamide
2-(cyclohexylmethyl)-4-(1H-imidazole-5-carbonyl)morpholine
{1-[1-(1-benzylpiperidin-4-yl)piperidin-3-yl]piperidin-4-yl}methanol
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(methylamino)pyridine-3-carboxamide
1-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)-3-phenoxypropan-1-one
(4-{[4-(5-methylfuran-2-yl)phenyl]methyl}morpholin-2-yl)methanamine
3-[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)methyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{5-[1-(4-methyl-1H-pyrazol-1-yl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
2-{[4-(3-methoxyphenyl)-5-(4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
methyl 5-{[(2,4-dimethoxyphenyl)methyl]amino}-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(5-methylfuran-2-yl)methyl]-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-benzyl-5-(1H-indazole-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[2-(4-methanesulfonylphenyl)-4-methylphenoxy]acetamide
2-(1-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-(4-cyanopyridin-2-yl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
2-[4-(2,2-dimethylpropyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-(furan-3-ylmethyl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(5-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3S)-1-benzylpyrrolidin-3-yl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
[(2,5-dimethylphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
3-(2-methyl-1H-1,3-benzodiazol-6-yl)-1-[2-(piperidin-1-yl)ethyl]urea
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(3-methylpyridin-2-yl)piperazine
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine