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(2S)-4-methyl-2-phenyl-1-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
2-(3-methylbut-2-en-1-yl)-8-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1λ6-thiomorpholine-1,1-dione
N-[(4-fluorophenyl)methyl]-3-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-4-yl)propanamide
3-{[2-(2-amino-1,3-thiazol-4-yl)ethyl]sulfamoyl}-N-ethyl-N-methylbenzamide
{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}[(2,2-dimethyloxan-4-yl)methyl]amine
N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-1,3-thiazole-5-carboxamide
1-phenyl-N-[(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)methyl]methanesulfonamide
3-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
2-(2H-1,3-benzodioxol-5-yl)-N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)acetamide
1-(3-{3-[(4-benzylpiperidin-1-yl)methyl]phenoxymethyl}piperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
7-(cyclopropylmethyl)-2-[4-(1H-imidazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
methyl (2S,4S)-4-[2-(4-methoxy-3-methylphenyl)acetamido]-1-methylpyrrolidine-2-carboxylate
1-(3-methoxypropyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
2-(dimethylamino)-7-(2,2-diphenylacetyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-({4-[4-methyl-2-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
methyl 4-[3-(2-phenylacetyl)piperidine-1-carbonyl]benzoate
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(4-methyl-1H-imidazol-5-yl)methyl]amine
(1S,5R)-6-(pyridin-2-ylmethyl)-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{imidazo[1,2-a]pyridin-3-yl}-N-[(2-methoxyphenyl)methyl]-N-propylacetamide
(1S,5R)-6-(4-ethylbenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
methyl[2-(1-methylpiperidin-4-yl)ethyl][(3-methylthiophen-2-yl)methyl]amine
N5-cyclohexyl-1-cyclopropyl-N3-methyl-4-oxo-N3-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-5-(trifluoromethyl)pyridine
8-{[3-(trifluoromethoxy)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}-5-cyclopropyl-1,2-oxazole
3-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(morpholin-4-yl)ethyl]benzamide
(3R,4S)-1-[4-(2-methoxyphenyl)benzoyl]-4-propylpyrrolidin-3-amine
6-(3-oxo-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propyl)-2,3-dihydropyridazin-3-one
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-4-phenyl-N-(pyridin-3-ylmethyl)benzamide
1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carboxylic acid
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-(dimethylamino)-N-(2-hydroxyethyl)acetamide
N-(furan-2-ylmethyl)-4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
dimethyl[3-(3-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}phenoxy)propyl]amine
1-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperidine-4-carboxylic acid
N-({1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
2,2-dimethyl-N-(1-{1-[1-(6-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
1-cyclohexyl-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-pyrazol-5-yl)acetamide
2-(furan-2-yl)-N-({1-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-yl}methyl)-2-oxoacetamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-(cyclohex-3-ene-1-carbonyl)-6-methyl-5-[5-(3-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
methyl 2-{[(2-methoxyphenyl)methyl](propyl)carbamoyl}benzoate
1-(2-methoxypyridine-4-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane