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3-phenyl-N-(1-{7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
1-(2-aminoethyl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(1H-imidazole-2-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
5-methyl-3-(oxan-4-yl)-1-{[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-1,2,4-triazole
1-[1-(2-aminoethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-N-ethylpiperidine-1-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
(4aR,8aR)-6-[(2E)-3-phenylprop-2-en-1-yl]-1-(2,3,4-trifluorobenzoyl)-decahydro-1,6-naphthyridine
3-{[(cyclohexylmethyl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
5-{[(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]methyl}-1,2,4-oxadiazole-3-carboxamide
(4aS,7aR)-1-(5-fluoro-2-methylbenzoyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[4-(3-methoxypyrazin-2-yl)phenyl]methanol
N-[1-ethyl-2-(2-fluorophenyl)-7-(4-methoxypiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-(oxan-2-ylmethyl)acetamide
4-{5-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(5-chlorothiophene-2-carbonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-{6-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridin-3-yl}ethan-1-one
(1R,2R,4R)-N-[(dimethyl-1,3-thiazol-2-yl)methyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(1-propylpiperidin-4-yl)propanamide
3-[(2R,3R,6R)-5-[(5-methylthiophen-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
methyl 4-[({2-[5-oxo-1-(2-phenylethyl)pyrrolidin-2-yl]ethyl}amino)methyl]benzoate
N-methyl-5-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-[(3R,4S)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-ethyl-N-(2-hydroxyethyl)-5-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
1-[2-(trifluoromethyl)morpholine-4-carbonyl]naphthalen-2-ol
4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1λ6-thiomorpholine-1,1-dione
N-[(5-chloro-1H-indol-2-yl)methyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(pyrazin-2-ylmethyl)acetamide
4-(5-chloro-3-fluoropyridin-2-yl)piperazine-2-carboxylic acid
diethyl({2-[5-(2-methyl-1,3-thiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl})amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]propanamide
5-chloro-2-oxo-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-3-carboxamide
4-amino-2-(morpholin-4-yl)-5-[2-(propan-2-yl)pyrimidin-4-yl]-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
2-(4-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
1-(3,5-dimethylphenyl)-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-2-one
1-[(2-chlorophenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(2-aminopyridine-4-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
1-[(3-chloropyridin-4-yl)methyl]-3-phenylpyrrolidin-3-ol
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one