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N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]oxolane-2-carboxamide
N-ethyl-5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrimidin-2-amine
3-[(4-methoxy-4-phenylpiperidin-1-yl)methyl]-7-methyl-1,2-dihydroquinolin-2-one
2-{5-[2-(2-hydroxyethoxy)phenyl]-4-phenyl-1H-imidazol-1-yl}acetic acid
7-(5-methylthiophen-2-yl)-4-(1H-pyrazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-1H-indole
N-methyl-5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyrimidin-2-amine
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
3-{5-[2-methyl-2-(morpholin-4-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-(pyridin-2-ylmethyl)urea
N-[(3-methylphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
[(4-fluorophenyl)methyl]({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(pyridin-4-ylmethyl)amine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-4-(1H-pyrazol-3-yl)benzamide
2-ethoxy-3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}pyridine
N-(5-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonane-7-carbonyl}-1,3-thiazol-2-yl)acetamide
ethyl 1-(2-oxo-2-phenylacetyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
methyl 5-[(2-methylpropyl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{2-hydroxy-3-[2-methoxy-4-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-(trifluoromethyl)benzamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(2,3-dihydro-1H-isoindol-2-yl)propan-1-one
ethyl N-{2-oxo-4-[3-(1H-pyrazol-1-yl)phenyl]-1,2,3,4-tetrahydroquinolin-7-yl}carbamate
4-[(dimethylamino)methyl]-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}azepan-4-ol
5-(azocane-1-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
3-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridin-2-ol
(1R,5R)-6-(3,5-difluoropyridine-2-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
4-{butyl[2-(1-methylpiperidin-4-yl)ethyl]amino}butan-1-ol
(3aR,6aR)-2-[4-(hydroxymethyl)benzoyl]-5-(3-methylbut-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl (2S)-2-{[7-acetyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-2-cyclopropylacetate
5-phenyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-pyrrole-2-carboxamide
4-[2-(2,3-dimethylphenoxy)ethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{1-oxo-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]propan-2-yl}methanesulfonamide
methyl 2-[(4-methylphenyl)sulfamoyl]-6-(pyrazine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[3-(2H-1,3-benzodioxol-5-yl)propyl]pyridine
5-(2-chloro-6-methoxyphenyl)-2,4-dimethyl-1,3-thiazole
1-ethyl-5-oxo-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrrolidine-3-carboxamide
1-[(3-{[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N,N-dimethyl-2-{[(2-methyloxolan-2-yl)formamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
methyl (2S)-3-methyl-2-[(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}phenyl)formamido]butanoate
6-[4-(hydroxymethyl)-4-(oxan-2-ylmethyl)piperidin-1-yl]pyrazine-2-carboxamide
(1S,5R)-3-[2-(4-fluorophenoxy)ethyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{[(5,6-dimethylpyrimidin-4-yl)amino]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyrimidin-4-yl)pyrrolidin-3-ol
9-[(4-chlorophenyl)methyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(4-methyl-1,3-thiazol-5-yl)-1H-pyrazol-1-yl]-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]propanamide
1-(1-cyclohexylpiperidin-3-yl)-4-(4-fluorophenyl)piperazine
2-ethyl-9-[2-(4-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{[(4-chlorophenyl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol