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methyl 6-(cyclopent-1-ene-1-carbonyl)-2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl (2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-4-(cyclopropylmethyl)piperidine-4-carboxylic acid
1-(2-methyl-4-phenylpiperazin-1-yl)-3-(1H-pyrrol-1-yl)propan-1-one
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}amine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-methyl-1H-imidazole-4-sulfonamide
1-(2-methylphenyl)-4-[2-(pyridin-3-yl)acetyl]piperazin-2-one
2-(4-chloro-3-fluorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(2-methylphenoxy)ethan-1-one
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
6-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
6-(3,5-dimethylphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
6-(5-methyl-1H-pyrazole-3-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
ethyl 1-(1-benzylpiperidin-4-yl)-4-(cyclopropylmethyl)piperidine-4-carboxylate
1-[3-(2-methoxybenzamido)phenyl]-5-oxopyrrolidine-3-carboxylic acid
1-ethyl-3-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-1-benzofuran-3-carboxamide
2-{2-[1-(7-chloroquinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
5-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
2-(4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}morpholin-2-yl)ethan-1-ol
N-[2-methyl-2-(morpholin-4-yl)propyl]-2-oxo-2-(thiophen-2-yl)acetamide
(2S,4R)-N,N-diethyl-1-methyl-4-(4,5,6,7-tetrahydro-1-benzothiophene-2-amido)pyrrolidine-2-carboxamide
N-benzyl-5-(2,4-difluorophenoxymethyl)-N-ethyl-1,2-oxazole-3-carboxamide
4-(2-chlorophenoxy)-1-(oxolan-3-ylmethyl)piperidine
1,2-dimethyl-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
N-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5-ethyl-4-({4-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)furan-2-carboxamide
4-(7-fluoro-2-methylquinoline-4-carbonyl)piperazin-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(naphthalen-2-yl)piperazin-1-yl]propan-1-one
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-methyl-1,4-diazepan-5-one
4-(2-oxopyrrolidin-1-yl)-N-(1-phenylbutyl)benzamide
(4aS,7aR)-1-(2-methoxy-5-methylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
3-[2-(piperidin-2-yl)ethyl]-5-(pyridin-3-yl)phenol
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
1-(3-fluoro-2-methylbenzoyl)-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepan-6-ol
1-[2-(dimethylamino)ethyl]-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
2-(1-{[1-(1-methylcyclopropanecarbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
6-ethyl-2-methyl-N-(oxan-3-yl)quinoline-4-carboxamide
(3S,4S)-1-[(2,5-dimethylphenyl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
4-(2-methylquinolin-6-yl)-1-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]piperidin-4-ol
2-(2H-1,3-benzodioxol-5-yloxy)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}acetamide
2-cyclopropyl-8-[2-(2-methoxy-4-methylphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(2-fluoroethyl)-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetamide