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1-[2-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
2-amino-4-(6-methylquinolin-5-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1-ethyl-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1H-pyrazole-4-carboxamide
2-[5-(5-ethyl-1,3-oxazol-4-yl)-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-3-yl]acetamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(2-methylprop-2-en-1-yl)piperidine-3-carboxamide
2,5-dimethoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-[(3R,4R)-3-hydroxy-1-(3-methoxypyrazin-2-yl)piperidin-4-yl]pyridine-2-carboxamide
4-{1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-phenyl-1H-pyrazole
5-{[benzyl(methyl)amino]methyl}-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-1,2-oxazole-3-carboxamide
N-methyl-4-(2-methyl-1H-imidazol-1-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
1-{1-[6-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-2-(pyridin-3-yl)morpholine
1-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1-methylcyclohexane-1-carboxamide
5,8-dimethoxy-4-methyl-2-[2-(trifluoromethyl)morpholin-4-yl]quinoline
2-methoxy-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-sulfamoylbenzamide
(3S,4S)-4-cyclopropyl-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-phenyl-1,2-oxazole-3-carboxamide
8-fluoro-2-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)quinolin-4-ol
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-methylphenyl)-1H-pyrazole
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
(1S,5R)-N-[4-(methylsulfanyl)phenyl]-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-(thiophen-2-ylmethyl)acetamide
(2S,4R)-4-amino-1-[3-(2-oxoazepan-1-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxopentan-2-yl}acetamide
ethyl({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}-1H-indole
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
8-[(dicyclopropylmethyl)amino]-2,6-dimethyloctan-2-ol
N4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-6-(propan-2-yl)pyrimidine-2,4-diamine
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-2-carboxamide
N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-[(4-fluorophenyl)methyl]-4-(2-methyl-1,3-thiazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
5-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-[2-chloro-5-(morpholin-4-yl)phenyl]-1-[1-(pyrazin-2-yl)propan-2-yl]urea
8-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-aminoethyl)-5,6-dimethyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
2-{1-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}benzoic acid
4-(2-methoxyphenoxy)-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
1-(2-cyclohexylethyl)-3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-3-hydroxypiperidin-2-one
6-ethyl-3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(3-fluorophenyl)-3-{1-[1-(3-methylbutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
7-fluoro-2-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]quinoline-4-carboxamide
4-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(2-methoxyphenyl)-5-methyl-4-[3-(thiophen-3-yl)propanoyl]piperazin-2-one