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4-[(4-fluorophenyl)methyl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
8-{3-carbamoyl-5H,6H,7H-cyclopenta[b]pyridin-2-yl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
6-(2-methylphenyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}imidazo[2,1-b][1,3]thiazole
6-ethyl-2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-N-methyl-N-propylquinoline-4-carboxamide
N-[2-(3-methoxyphenyl)-1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}ethyl]-N-methylpyridine-2-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5-(3-methoxyphenyl)-N-methylfuran-2-carboxamide
5-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-{2-oxo-2-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethyl}-1,3-oxazolidin-2-one
(3S,4S)-4-cyclopropyl-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidine-3-carboxylic acid
1-(1H-indazol-5-yl)-4-{[4-(2-methylpropyl)phenyl]methyl}piperazin-2-one
N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-(4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[(2,4-dichloro-5-fluorophenyl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
1-{[(3R,4R)-1-(2-chloro-6-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[1-(1-methyl-1H-imidazol-2-yl)butyl]amine
1-[2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)pyrimidin-4-yl]pyrrolidin-3-ol
2-[4-(dimethylamino)phenyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
8-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
3-(1,3-benzothiazol-2-yl)-1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)propan-1-one
(1-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)(pyridin-2-yl)methanol
4-[(2-methylphenyl)methyl]-1-(2,5,7-trimethylquinoline-4-carbonyl)-1,4-diazepan-5-one
5-(cyclopropylamino)-N-[(2-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-methyl-2-({4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
(1R,3S)-7-(3-chlorothiophene-2-carbonyl)-3-[2-(dimethylamino)ethoxy]-7-azaspiro[3.5]nonan-1-ol
N-(isoquinolin-5-ylmethyl)-N-methyl-2,3-dihydro-1H-indene-1-carboxamide
N3-ethyl-4-oxo-1-(2-phenylethyl)-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(2-phenylethyl)piperazine
4-chloro-2-{[methyl({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amino]methyl}phenol
N-[(1-methylpyrrolidin-3-yl)methyl]-2-(pyridin-3-yloxy)acetamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidine
methyl 2-[(4-cyclopentylpyrimidin-2-yl)(methyl)amino]acetate
N-cyclopropyl-1-[(1s,4s)-4-(3-methylbenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(2-chlorophenyl)methyl]-6-(2-methylpropyl)-2-oxo-N-(propan-2-yl)-1,2-dihydropyrimidine-4-carboxamide
4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine
3-({4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridin-2-amine
(3R,5R)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
7-(cyclopropylmethyl)-2-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2,7-diazaspiro[4.5]decane
[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
8-methoxy-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carboxylic acid
1-benzyl-3-{2-[3-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-{3-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-(3-{1-[2-(1-methylpiperidin-2-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
2-{1-benzyl-4-[(2,3-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(dimethylamino)ethyl]-2,4-difluoro-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)benzamide