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1-(2-fluorophenyl)-4-[4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]piperidin-4-ol
N-{4-[(2,6-dimethylphenyl)carbamoyl]phenyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
7-(cyclobutylmethyl)-2-[2-(thiophen-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}ethan-1-one
methyl (2S,4R)-4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxylate
6-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
methyl 2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
(3R,4R)-1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-{4-[(dimethylamino)methyl]phenyl}pyridine-3-carboxylic acid
(3S,4S)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-(1-benzofuran-3-carbonyl)-4-(1H-imidazol-2-yl)piperidine
1-methyl-N-{[2-(5-methylfuran-2-yl)phenyl]methyl}-1H-1,2,3-triazol-4-amine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-propyl-1,3-thiazole-4-carboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(1,2-oxazol-5-yl)-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
2-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}pyridine-3-carboxamide
1-(5-chloro-2-fluorobenzoyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
5-methyl-4-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-(4-methylphenyl)piperazin-2-one
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
methyl 3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(3,5-dichloro-4-methylbenzoyl)piperidine-3-carbonitrile
N-(2,4,5-trifluorophenyl)-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[3-(pyridin-2-yl)propyl]carbamoyl}pyrrolidine-2-carboxylate
4-(5-methyl-1,3-oxazole-4-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[2-(5-methylfuran-2-yl)phenyl]methyl})amine
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
4-[1-(5-methanesulfonyl-2-methylpyrimidin-4-yl)piperidine-4-carbonyl]morpholine
1-benzyl-N,N-dimethyl-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(3,6-dimethylpyrazin-2-yl)-N,N-bis(propan-2-yl)benzamide
8-{[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
4-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}-2,6-dimethylphenyl acetate
ethyl 4-[(4-methoxyphenyl)methyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxylate
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
N-{2-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]ethyl}-3-methylpyridin-4-amine
6-[2-(2-chloro-4-fluorophenyl)acetyl]-N-(3,5-dimethylphenyl)-6-azaspiro[2.5]octane-1-carboxamide
N,2-dimethyl-N-[2-(oxan-2-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(3R,4R)-1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-fluoro-5-sulfamoylbenzamide
2-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-1,3-benzothiazole
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]quinoxaline
4-(azepan-1-yl)-5-methyl-N-[(5-methylfuran-2-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
4-[(4-ethoxyphenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
5-methoxy-1-methyl-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-indole
2-{4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]phenyl}acetic acid
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-3-(hydroxymethyl)piperidin-3-ol