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N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-oxo-N-phenylacetamide
7-(1,3-benzothiazol-2-yl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 2-[(1-ethyl-1H-imidazol-5-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
N-[(2R,3R)-2-ethoxy-1'-(5-methylpyrazine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
5-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
N-ethyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
1-(3-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-3,5-dimethyl-1H-pyrazole
5-[2-oxo-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-4-yl]thiophene-2-carboxylic acid
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(4-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-{2-[4-(1H-pyrazol-1-yl)phenyl]pyrimidin-4-yl}piperidin-3-ol
5-[4-hydroxy-1-(thiophen-3-ylmethyl)piperidin-4-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
9-[2-(2-fluorophenyl)acetyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N,1-dimethyl-N-[4-(morpholin-4-yl)butyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(oxan-4-yl)-2-(propane-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
3-{4-[6-(cyclopentylamino)pyridazin-3-yl]phenyl}propanoic acid
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazin-2-amine
9-ethyl-1-methyl-4-[3-(pyridin-4-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{4-[3-(propan-2-yloxy)phenyl]-1H-pyrazol-1-yl}propanamide
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
2-{[(3aS,6aS)-1-[(5-methylthiophen-2-yl)methyl]-octahydropyrrolo[2,3-c]pyrrol-5-yl]methyl}-5-(furan-2-yl)-1,3,4-oxadiazole
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
5-(1H-indol-1-ylmethyl)-N-[2-(propan-2-ylsulfanyl)ethyl]-1H-pyrazole-3-carboxamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide
methyl[3-(5-methylfuran-2-yl)butyl](1H-pyrazol-3-ylmethyl)amine
methyl 2-({1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-4-(methylsulfanyl)butanoate
N,N-dimethyl-2-[(1S,5R)-6-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-(4-chlorophenyl)-5-{1-[1-(1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
5-ethyl-2-{1-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-imidazol-2-yl}pyridine
(1S,2R)-2-[methyl({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amino]cyclohexan-1-ol
2-{1-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}pyridine
2-methoxy-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyridine-3-carboxamide
6-(2,3-dihydro-1H-isoindole-2-carbonyl)-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
8-fluoro-2-{[(1,3-thiazol-2-ylmethyl)amino]methyl}quinolin-4-ol
2-(oxolan-2-ylmethyl)-9-(1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydroquinoxalin-2-one
5-[1-(4-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1-(prop-2-en-1-yl)piperidin-2-one
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)ethan-1-one
7-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-[2-(1H-imidazol-1-yl)ethyl]-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(3S,4S)-3-[({3-[(4-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
3-{5-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridazine
2-methyl-8-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-2,8-diazaspiro[5.5]undecane
4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-3-(thiophen-2-yl)-1H-pyrazole
(1S,4S)-5-(2-hydroxyethyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane