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N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)propanamide
methyl N-{2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}carbamate
N-cyclopropyl-3-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]propanamide
1-[3-(diethylamino)pyrrolidin-1-yl]-3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(1-hydroxypropan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(5-methyl-4-{[3-(5-methyl-1H-pyrazol-1-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]-3-phenoxypropanamide
(3S,4R)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-ethyl-4-methylpiperidin-4-ol
2-(2,4-difluorophenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
4-[4-(ethanesulfonyl)piperazin-1-yl]-6-methyl-2-propylpyrimidine
3-(morpholin-4-yl)-N-[(2-phenoxypyridin-3-yl)methyl]propanamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-{4-[4-chloro-2-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
(3R,4R)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-{[5-(cyclohexylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,3-dimethylurea
N-(4-chloro-3-methoxyphenyl)-2-{[1-(furan-2-carbonyl)piperidin-3-yl]amino}acetamide
2-{3-[(3-chlorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-2-azabicyclo[2.2.1]heptane
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-3-yl)pyridine
6-[(2-fluorophenyl)methoxy]-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
5-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-methylazepane-2-carboxamide
1-(4-methoxyphenyl)-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclopentane-1-carboxamide
2-[1-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
2-{2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}-1,2,3,4-tetrahydroisoquinoline
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S)-3-ethyl-N-[(1R)-1-(4-methoxyphenyl)ethyl]morpholine-4-carboxamide
3-[({2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}amino)methyl]pyrrolidin-3-ol
3-(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-1,3-oxazolidin-2-one
2-{3-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
2-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1-methylpiperidine
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-3-(pyridin-3-yl)propan-1-one
1-cyclopentanecarbonyl-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
N-ethyl-N-methyl-6-[4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
2-methyl-5-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)-N-methylpyridin-2-amine
1-(2,5-dimethylfuran-3-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-(4-methylphenyl)-5-(pyridin-4-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrimidin-2-amine
5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-2-(piperidin-1-yl)pyrimidine
ethyl 3-[(2-methylphenyl)methyl]-1-(pyrazine-2-carbonyl)piperidine-3-carboxylate
1-[2-({furo[3,2-c]pyridin-4-yl}amino)ethyl]pyrrolidin-2-one
2-({4-[6-(1H-imidazol-1-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
1-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)piperazine
(3S,4R)-4-(4-fluorophenyl)-1-(2-propoxyethyl)pyrrolidine-3-carboxylic acid
1-[(2,2-dimethyloxan-4-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-amino-8-[3-(4-methoxyphenoxy)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-[(2,3-dimethoxyphenyl)methyl]-N-ethyl-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
7-[(2,3-dimethoxyphenyl)methyl]-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-{1-[(6-fluoroquinolin-2-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide