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5-{5-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
(1R,5R)-6-[5-(ethylsulfanyl)thiophene-2-carbonyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-cyclopentyl-4-[4-({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]benzamide
1-(4-methylbenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-5-methoxybenzoic acid
N-(2,4-dimethylphenyl)-2-({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}amino)acetamide
7-methoxy-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{1-benzyl-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-cyclopropyl-5-(2-hydroxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
5-methyl-1-{2-[3-(2-methyl-1,3-thiazol-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
N-methyl-2-(4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperazin-1-yl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
(3R,4S)-4-(5-methylfuran-2-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-3-amine
4-[(3-chlorophenyl)methyl]-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-phenylpiperazin-2-one
2-(4-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-N-ethylacetamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
3-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}propanamide
ethyl(2-methylprop-2-en-1-yl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-[3-(pyridin-2-yl)phenyl]urea
4-{1-[2-(diethylamino)acetyl]piperidin-3-yl}benzoic acid
4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1-methylimidazolidin-2-one
3-{[4-(2-phenylpyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
(2S)-2-({[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]carbamoyl}amino)-4-methylpentanamide
4-({1-[4-(4-methylphenyl)phenyl]piperidin-4-yl}amino)butan-1-ol
1-cyclohexyl-3-hydroxy-4-(1H-imidazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
8-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-8-azaspiro[4.5]decane-7,9-dione
2,6,6-trimethyl-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-1-propyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-{1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
2-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
2-methyl-5-{[3-(4H-1,2,4-triazol-4-yl)propyl]sulfanyl}-1,3,4-thiadiazole
2-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1λ6-thiolane-1,1-dione
2-ethyl-1-methyl-4-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
3-{1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}morpholine-2-carboxamide
3-(azepane-1-carbonyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
4-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
2-methyl-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-2-(thiophen-2-ylformamido)propanamide
1-ethyl-5-methyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
5-methyl-3-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-3,4-dihydroquinazolin-4-one
N-cyclopropyl-1-[(1s,4s)-4-(2-chlorobenzenesulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethyl)pyridine
1-[3-(dimethylamino)phenyl]-3-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}urea
4-(2,5-dimethoxybenzoyl)-3,4-dihydro-2H-1,4-benzoxazine
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-ethyl-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]urea