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4-methyl-2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole
6-fluoro-2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}quinolin-4-ol
(3R,4R)-1-[(4-chlorophenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
6-methyl-4-(2-methylpyrrolidine-1-carbonyl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline
5-(4-methoxyphenyl)-3-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-1,2,4-triazine
3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
1-({4-methyl-5-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-[(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,2-dimethylpiperazine
4-{4-[3-(methoxymethyl)piperidine-1-carbonyl]phenoxy}-N,N-dimethylpiperidine-1-sulfonamide
1-[3-(4-fluorophenyl)benzoyl]-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepan-5-one
3-(2-chloropyridin-3-yl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]urea
(4aS,8aR)-1-(2-aminoethyl)-6-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(pyridin-3-yl)piperidin-4-ol
5-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)benzonitrile
N-ethyl-4-methoxy-N-[1-(4-methoxyphenyl)propyl]cyclohexane-1-carboxamide
1-[3-(cyclopentyloxy)phenyl]-3-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]urea
1-(butan-2-yl)-N3-(furan-2-ylmethyl)-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[(3-chlorophenyl)methyl]-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1,3-benzoxazole-6-carboxamide
(butan-2-yl)(1H-imidazol-4-ylmethyl)(pyridin-3-ylmethyl)amine
3-cyclopropyl-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
8-methyl-5-[1-(2-phenoxyethyl)-1H-1,2,3-triazol-4-yl]quinoline
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-(2,3-dihydro-1H-inden-1-yl)-1,2-oxazole-3-carboxamide
4-methyl-2-[2-(trifluoromethyl)morpholin-4-yl]quinoline
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]furan-2-carboxamide
N,N-dimethyl-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidin-3-amine
7-(cyclopropylmethyl)-2-{2-[4-(hydroxymethyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}acetamide
(3R,4S)-4-cyclopropyl-1-[1-(2-methylphenyl)piperidin-4-yl]pyrrolidin-3-amine
N-(dimethyl-1,2-oxazol-4-yl)-4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}benzamide
N-(3-acetamidophenyl)-4-[(3-hydroxy-3-methylpiperidin-1-yl)methyl]benzamide
N-methyl-5-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-methylpyridin-4-yl)-4-[4-(piperidin-3-yl)benzoyl]-1,4-diazepane
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[cyclopropyl(pyridin-2-yl)methyl]-N-methyl-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-[3-({3-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[3-(dimethylamino)piperidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
N-(5-acetyl-2-ethoxyphenyl)-4-(4-fluorophenyl)piperazine-1-carboxamide
9-methoxy-3-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(1R,5S)-6-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
[3-benzyl-1-(2,4-difluorobenzenesulfonyl)piperidin-3-yl]methanol
N-cyclopropyl-3-{5-[3-(thiophen-3-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
7-{[benzyl(methyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}bis(1,3-oxazol-4-ylmethyl)amine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(isoquinolin-5-ylmethyl)methylamine