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4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperidin-4-ol
1-(4-methoxyphenyl)-5-[1-(pyrrolidin-1-yl)propyl]-1H-1,2,4-triazole
N-{[3-(2-methoxyethoxy)phenyl]methyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
2-[1-(1-methylpiperidin-4-yl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-2-yl]ethan-1-ol
1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-methylpent-3-en-1-yl)pyrrolidin-3-yl]-2,4-dimethylpyrimidine-5-carboxamide
N-(2-methoxyethyl)-1-(3-methylbutyl)-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}morpholine
1-(4-methoxybenzoyl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
2-[1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]benzoic acid
N-benzyl-1-(4,7-dimethylquinazolin-2-yl)piperidine-3-carboxamide
6-{3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
1-(4-fluorophenyl)-4-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]piperazine
(3S,7S,8aS)-7-{[(3-fluorophenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
(2R)-N-[4-(5-methylfuran-2-amido)phenyl]-5-oxopyrrolidine-2-carboxamide
ethyl 4-[3-(phenylamino)piperidin-1-yl]piperidine-1-carboxylate
methyl 5-[(2,2-dimethylpropyl)amino]-3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-methyl-4-phenyl-N-[2-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
1-(4-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(propan-2-yl)propanamide
4-fluoro-N-[2-(2-methoxy-5-{[methyl(propan-2-yl)amino]methyl}phenoxy)propyl]benzamide
8-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(3S,4R)-4-(2-methoxyphenyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
4-{4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrimidin-2-amine
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-{[4-(propan-2-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-ethyl-3-{1-[3-(2-oxoimidazolidin-1-yl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(pyridin-3-ylmethyl)-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-ethyl-1-methyl-3-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-2-(methylamino)-N-(prop-2-en-1-yl)pyridine-4-carboxamide
9-[2-(methylamino)acetyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-[3-(pyridin-2-yl)propyl]acetamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]piperidin-4-amine
S-{4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]phenyl}-2-hydroxy-N-methylethane-1-sulfonamido
3-benzyl-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
4-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}methyl)hepta-1,6-dien-4-ol
2-(5-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
1-(oxolane-3-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}pyridine-4-carboxamide
4-(5-methylpyridin-2-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-4-ol
5-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-(1H-1,2,3-triazole-5-carbonyl)-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine