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1-[2-(4-fluoro-2-methylphenyl)acetyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
3-(2-amino-4-{[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}-6-methylpyrimidin-5-yl)propanoic acid
(2S,4R)-4-amino-1-[2-(3-ethyl-2-imino-2,3-dihydro-1H-1,3-benzodiazol-1-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-cyclopropyl-6-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
4-{[2-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}-1,5-dimethyl-1H-pyrazole
2-(3-chloro-5-fluorobenzoyl)-6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrimidin-2-amine
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-fluoro-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1'-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-(naphthalene-1-carbonyl)piperidine
N-(1-carbamoylcyclopentyl)-4-(cyclobutylsulfamoyl)benzamide
N-(3,4-dimethoxyphenyl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-amine
1-(2,6-dimethylpyridin-4-yl)-4-(thiophen-3-ylmethyl)piperazine
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(cyclohexylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){2-phenyl-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]ethyl}amine
4-cyano-N-[2-(cyclohex-1-en-1-yl)ethyl]-1-methyl-N-[(4-methylphenyl)methyl]-1H-pyrrole-2-carboxamide
N-(pyridin-2-ylmethyl)-4-(1,3-thiazol-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-(3-methoxypropyl)-1-(2-methyl-1-benzofuran-7-carbonyl)piperidine
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(5-methyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-{[3-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyridine
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-ethyl-9-[4-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N,1-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-indole-3-carboxamide
1-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)ethan-1-one
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)pyridine-2-carboxamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methylthieno[3,2-d]pyrimidin-4-amine
(3E)-1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]hex-3-en-1-one
9-(3,5-dichloropyridin-2-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-hydroxy-N-{[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-4-methoxybenzamide
9-methoxy-3-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzene-1-sulfonamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(thiophen-2-yl)propanoyl]piperidine-4-carboxylic acid
3-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-methyl-1,2-dihydropyridin-2-one
4-hydroxy-N-[(2-methoxyphenyl)methyl]-N-(3-methoxypropyl)-2-methylpyrimidine-5-carboxamide
methyl 1-[1-ethyl-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carbonyl]piperidine-2-carboxylate
4-[(2-methylpyridin-3-yl)oxy]-N-[1-(pyridin-3-yl)propyl]piperidine-4-carboxamide
(3S,4R)-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(1S,5R)-6-(cyclopropylmethyl)-3-[(5-ethylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(3aR,6aR)-2-cyclohexyl-5-(2-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-chloro-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}imidazo[2,1-b][1,3]thiazole
1-methyl-N-[2-(pyridin-4-yl)ethyl]-1H-indole-6-carboxamide
2-methyl-4-phenyl-5-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
2-[(2-hydroxyethyl)({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
3-[2-(3-fluorophenyl)acetyl]-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(2,3-dihydro-1H-inden-2-yl)piperazine
(3S,4S)-3-({2-cyclopentyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}amino)-4-hydroxy-1λ6-thiolane-1,1-dione
2-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one