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N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
5-methoxy-1-methyl-N-[2-(quinolin-8-yloxy)ethyl]-1H-indole-2-carboxamide
(1S,5R)-3-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1'-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
8-[(3-chlorophenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-2-cyclopentanecarbonyl-5-(2-phenoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-{[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)acetamide
3,4,4-trimethyl-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)benzoyl]pyrrolidin-3-ol
2-{2-methyl-6-[4-(4-methylphenoxy)piperidin-1-yl]pyrimidin-4-yl}ethan-1-amine
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-ol
N-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]quinoline-4-carboxamide
1-(3,5-dimethylphenyl)-4-(2-methoxypyridine-4-carbonyl)piperazin-2-one
N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-1H-indazole-3-carboxamide
1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[2-(piperazin-1-yl)ethyl]piperidin-4-amine
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
7-methanesulfonyl-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(2-methoxyethyl)(methyl)amino]-1-[4-(4-methylphenoxy)piperidin-1-yl]ethan-1-one
2-methyl-6-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
1-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methylpiperazine
1-(4-{4-chloro-2-[2-(2-hydroxyethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methylbut-2-en-1-yl)piperidine
3-chloro-6-methyl-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyrazolo[1,5-a]pyrimidine
1-[(6-methylpyridin-2-yl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methoxybenzoyl)piperidine
2-(3-methoxypropyl)-8-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-N-[1-(4-methylphenyl)-5-oxopyrrolidin-3-yl]-1H-indole-6-carboxamide
(2E)-3-(pyridin-2-yl)-1-(4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)prop-2-en-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
(4aS,8aR)-6-[2-(benzyloxy)acetyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
5-{2-[(2-methoxyethyl)amino]ethyl}-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
(2E)-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-3-phenylprop-2-enamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-fluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-hydroxy-3-{[methyl(thiophen-2-ylmethyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
1-(2,3-dimethylphenyl)-N-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-hydroxy-2-[(phenylsulfanyl)methyl]-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidine-5-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)benzamide
N,N-dimethyl-2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)acetamide
4-[3-cyclopropyl-1-(4-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]-2-methyl-1,2-dihydrophthalazin-1-one
(1R,5R)-6-(cyclobutylmethyl)-3-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-(dimethylamino)propyl]-9-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-3-(piperidin-4-ylmethyl)benzamide
2-{4-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
2-({4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
1-[(4-fluorophenyl)methyl]-5-[2-(pyridin-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-(2-{1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]piperidin-2-yl}ethyl)phenol
1-[(diethylcarbamoyl)methyl]-N-(1-hydroxy-3-methylbutan-2-yl)-1H-1,2,3-triazole-4-carboxamide