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1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-methanesulfonamidopropanamide
5-(4-benzoylpiperidine-1-carbonyl)-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
5-tert-butyl-4-{[(3S,4R)-3-cyclopropyl-4-acetamidopyrrolidin-1-yl]methyl}furan-2-carboxamide
(2S,4S)-4-amino-N-[(2,4-dichlorophenyl)methyl]-1-methylpyrrolidine-2-carboxamide
3-(naphthalene-1-carbonyl)-1-(3,4,5-trimethoxybenzoyl)piperidine
[(1,2-dimethyl-1H-imidazol-5-yl)methyl]({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amine
2-(1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
5-chloro-2-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
N-[(2-fluorophenyl)methyl]-4-[4-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)piperidin-1-yl]benzamide
2-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
5-(3-methoxyphenyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,2,4-triazin-3-amine
N-[3-(dimethylamino)-1-phenylpropyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{[1-(hydroxymethyl)-9-[3-(methylsulfanyl)propyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl}benzonitrile
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
5-{2-[(4-methoxyphenyl)methyl]morpholine-4-carbonyl}-2-methyl-1H-1,3-benzodiazole
(5-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
(3R,5R)-N-cyclohexyl-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carboxamide
9-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
1-(2,6-dimethylpyrimidine-4-carbonyl)-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
3-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-1-ium-1-olate
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-octahydropyrrolo[1,2-a]piperazine
(3aR,6aR)-2-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydroisoquinolin-1-one
5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N5-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
(1S,5R)-3-benzyl-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)methyl]-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-methyl-5-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrazine
6-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}quinoxaline
2-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-3-(thiophen-2-yl)propan-1-ol
4-({4-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1-(4-methoxyphenyl)-5-methyl-1H-pyrazole
2-(phenylsulfanyl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-(2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1-{7-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
5-acetamido-2-ethyl-N-[3-(morpholin-4-yl)propyl]-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
5-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}phenyl)-1H-1,2,4-triazole
3-(3-methoxyphenyl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
1-{4-[4-(azocane-1-carbonyl)phenoxy]piperidin-1-yl}-2-methoxyethan-1-one
1-(1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
4-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-3,3-dimethylpiperazin-2-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenylpropanamide
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4,4-difluoropiperidine
N-ethyl-5-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-benzofuran-2-carboxamide
2-[4-(pyridin-3-yloxy)piperidin-1-yl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidine
1-methyl-5-(4-methylpiperazin-1-yl)-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(2-chlorophenyl)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
2-cyclopropyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]quinoline-4-carboxamide