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2-(4-phenylmethanesulfonylmorpholin-3-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
(2S,4S)-4-amino-N-methyl-1-{2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}pyrrolidine-2-carboxamide
2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-4-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-{2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-4-fluorobenzamide
N-[2-(3-methoxyphenyl)phenyl]-1-(naphthalen-1-ylmethyl)piperidine-4-carboxamide
1-[2-(pyridin-2-yl)-4-{[2-(pyrrolidin-1-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
N2-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-5-fluoro-N4-methylpyrimidine-2,4-diamine
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
[(2,3-dimethyl-1H-indol-7-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-[3-(1H-indol-1-yl)propyl]-1-(pyrimidin-2-yl)piperidin-4-amine
1-cyclopropyl-4-[4-(2-methylphenoxy)piperidine-1-carbonyl]pyrrolidin-2-one
1-(3-methoxyphenyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-2-one
3-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[2-(trifluoromethoxy)phenyl]urea
4-(4-propyl-1H-1,2,3-triazol-1-yl)-1-(1-propylpiperidin-4-yl)piperidine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-yl]methanol
3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}cyclobutan-1-amine
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
N'-cycloheptyl-N-[2-methyl-2-(morpholin-4-yl)propyl]butanediamide
5-methoxy-2-({4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-ethyl-3-methylpiperidine-3-carboxamide
N-{[1-(2,2-dimethylpropyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]-2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazole
(3S,4R)-3-methoxy-1-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]piperidin-4-amine
N-(1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1H-indole
2-cyclopropyl-N-[(1R)-1-(4-fluorophenyl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-hydroxy-3-{[methyl(prop-2-en-1-yl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-sulfamoylbenzamide
2-[(3,5-difluorophenyl)methyl]-8-[(2R)-2-hydroxypropanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-3,4,7-trimethyl-1H-indole
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
1-(3,4-difluorophenyl)-5-(dimethyl-1,2-oxazol-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
4-[3-(propan-2-yloxy)benzoyl]piperazin-2-one
2-(3-methylbut-2-en-1-yl)-8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(2S,4R)-1-acetyl-4-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-amido}-N-ethylpyrrolidine-2-carboxamide
4-[(4-ethylphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3aR,6aR)-2-[1-(methoxymethyl)cyclobutanecarbonyl]-5-(pyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(3-methylphenoxy)ethan-1-one
N-(2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}ethyl)methanesulfonamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(2E)-3-(2-fluorophenyl)-N-{[3-methyl-7-(3-phenoxypropanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}prop-2-enamide
dimethyl(2-{[(4-methyl-1H-imidazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}ethyl)amine
N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-methylpyrimidin-2-amine
N-cyclopropyl-2-(thiophen-3-yl)pyridine-3-carboxamide
1-(oxan-4-yl)-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1,4-diazepan-6-ol