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N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
2-(azepan-1-yl)-N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)acetamide
8-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(2S)-2-(7-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyrrolidin-1-yl]ethan-1-one
3-[1-(2,5-difluorophenyl)cyclopropyl]-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-cyclopropyl-3-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]propanamide
1-[benzyl(methyl)amino]-3-{5-[(cyclopropylamino)methyl]-2-methoxyphenoxy}propan-2-ol
N-methyl-3-[methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl})amino]butanamide
N3-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(1S,6R)-N-(2-phenylphenyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
methyl[(1-methylpyrrolidin-2-yl)methyl][(2,3,4-trimethoxyphenyl)methyl]amine
7-(5-chloropyridin-2-yl)-4-(3-hydroxypropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]methanesulfonamide
2-(4-fluoro-3-methoxyphenyl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-[2-(2-ethoxyphenyl)ethyl]-4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
4-(3-cyanopyrazin-2-yl)-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]piperazine-1-carboxamide
1-(3-chlorophenyl)-4-(1H-pyrazole-3-carbonyl)piperazin-2-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetamide
[3-(2-methoxyethyl)-1-[1-(2-methylphenyl)piperidin-4-yl]piperidin-3-yl]methanol
1-[1-(1-benzofuran-3-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]oxolane-2-carboxamide
1-[(2,3-dichlorophenyl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
(4S,4aS,8aS)-4-phenyl-1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-decahydroquinolin-4-ol
1-(3-methoxypropanoyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
5-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
8-acetyl-2-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2,3,6-trimethyl-4-(3-phenoxyazetidine-1-carbonyl)quinoline
2-cyclopentyl-9-(6-cyclopropylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{[benzyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-2-(cyclopent-2-en-1-yl)ethan-1-one
2-{[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]amino}pyridine-3-carboxamide
5-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]-1,2-oxazole-3-carboxamide
({2-[(2-chlorophenyl)methoxy]-7-methoxyquinolin-3-yl}methyl)(1-methoxypropan-2-yl)amine
(1R,3S)-3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclopentan-1-amine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(pyridin-2-ylsulfanyl)propanamide
4-{[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[3-(2-chlorophenyl)phenyl]-2-methoxyacetamide
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]propanamide
N5-cyclooctyl-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-N3-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{2-[2-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-[1-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-4-oxo-4-phenylbutanamide
2-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidin-4-amine
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
(2E)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(pyridin-2-yl)prop-2-en-1-one
2-{3-[2-(4-chlorophenyl)morpholine-4-carbonyl]-5-methyl-1H-pyrazol-1-yl}-N-methylacetamide
N-methyl-6-oxo-1-(3-phenylpropyl)-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
2-[4-(hydroxymethyl)oxan-4-yl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 1-benzyl-5-(cyclobutylamino)-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methoxy-4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyridine