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5-(2-fluorophenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
[(2-butyl-1H-imidazol-4-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
(2S,4S)-N-ethyl-1-[(2E)-3-phenylprop-2-en-1-yl]-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-(4-methyl-1H-pyrazol-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
4-[4-(4-methoxyphenyl)-1H-imidazol-2-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(2-oxopiperidin-1-yl)acetamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
1-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-3-[4-(oxolan-2-yl)butyl]urea
2-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-imidazol-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
1-cyclopentyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-3-carboxamide
2,6-dihydroxy-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}benzamide
2-(1-{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-hydroxy-3-methylbenzamide
1-[(3-methoxyphenyl)methyl]-4-[5-oxo-1-(propan-2-yl)pyrrolidine-3-carbonyl]piperazin-2-one
2-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-{1-[({[1-(4-methoxyphenyl)cyclopentyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-2-(2-oxopiperidin-1-yl)acetamide
N-methyl-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
N-[3-(cyclopentyloxy)propyl]-5-methyl-2-phenyl-1H-imidazole-4-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylbenzamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[3-(phenylsulfanyl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-chloro-5-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
8-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
1-[(2,6-difluorophenyl)methyl]-3-(1-ethyl-1H-imidazol-2-yl)piperidine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1-methylcyclopropanecarbonyl)pyrrolidin-3-yl]-1-methyl-1H-imidazole-5-carboxamide
N-[2-hydroxy-2-(3-methoxyphenyl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(2,5-dimethoxyphenyl)-N-(furan-2-ylmethyl)-N-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}acetamide
N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-2-(morpholin-3-yl)acetamide
3-(1-ethyl-1H-imidazol-2-yl)-1-(2,3,4-trimethoxybenzoyl)piperidine
3-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3-diazinane-2,4-dione
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-chloropyrimidine
(3S,4R)-1-(1-acetylpiperidine-4-carbonyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
2-amino-4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-ethyl-1-[(8-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidine-3-carboxamide
2-(furan-2-yl)-7-methyl-N-(thiolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl[(5-propylfuran-2-yl)methyl](pyrazin-2-ylmethyl)amine
N-(pyridin-2-ylmethyl)-3-({1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-4-yl}oxy)benzamide
1-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-methyl-4-(4-{[4-(2-methylpropyl)piperazin-1-yl]methyl}phenyl)butan-2-ol
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-hydroxy-2-(pyridin-2-yl)ethyl]benzamide
6-fluoro-4-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 1-ethyl-5-{[(3-fluorophenyl)methyl]amino}-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(thian-4-yl)piperazine
1-{4-[2-(2,5-dichlorophenyl)-1H-imidazol-1-yl]butan-2-yl}-4-methylpiperazine
(1S,5R)-3-(4-fluorobenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one