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1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidin-4-amine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2,7-dioxo-1,3-diazepane-4-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-propanoylpiperidine-4-carboxamide
2-{4-[({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]piperidin-1-yl}ethan-1-ol
(2E)-3-(3-fluorophenyl)-1-{4-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}prop-2-en-1-one
N-[2-(2-fluorophenyl)ethyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
7-(2-hydroxyethyl)-2-{2-methylthieno[2,3-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
2-{[1,2,4]triazolo[4,3-a]quinolin-1-yl}-1,3-thiazole
2-{1-[(2-methylphenyl)methyl]-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(1H-pyrazol-1-yl)-1-[4-(pyridin-4-yl)piperidin-1-yl]butan-1-one
3-({4-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]phenyl}methyl)-5-methyl-4H-1,2,4-triazole
methyl 4-{3-[2-(cyclohexylformamido)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}benzoate
1-[4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
7-methyl-3-[(5-oxo-1,4-diazepan-1-yl)methyl]-1,2-dihydroquinolin-2-one
3-methyl-1-phenyl-5-(2,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
2-[({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}(methyl)amino)methyl]-3,4-dihydroquinazolin-4-one
N-[1-(1H-1,2,4-triazol-5-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
3-{1-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-[(3S,4R)-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-(4-ethoxy-2-fluorophenyl)-3-methyl-3-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]urea
4-(2,3-dimethyl-1H-indole-7-carbonyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}acetamide
butyl N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-N'-(2,4,6-trimethylphenyl)butanediamide
5-[(2E)-but-2-en-1-yl]-N-methyl-N-[(2-methylpyridin-4-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
9-(2-hydroxy-4-methylbenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-(2-aminopyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-methanesulfonylpropanamide
2-{[5-(furan-2-yl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(1S,6R)-9-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
4,6-dimethyl-5-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-1H-pyrazolo[3,4-b]pyridin-3-amine
4-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}benzoic acid
3-(3-chlorobenzoyl)-N-(4-fluorophenyl)piperidine-1-carboxamide
N-benzyl-N-(2-hydroxyethyl)-3-propanamidobenzamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-methoxy-1-methyl-1H-indole-2-carboxamide
8-[2-(cyclopentyloxy)phenyl]-2-(dimethylamino)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-[(3S,4R)-1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
5-(2H-1,3-benzodioxol-4-yl)-1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazole
N-cyclopentyl-2-({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}amino)propanamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-[(4-fluorophenyl)formamido]propanamide
N-cyclopropyl-2-(2,5-dimethylphenoxy)-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanamide
4-ethyl-3-{1-[4-(1H-indol-3-yl)butanoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridine-3-carboxamide
{[3-(azepan-1-yl)propyl](methyl)sulfamoyl}(benzyl)amine
1-(4-{2-[(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}urea
6-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)pyridine-2-carbonitrile
4-{1-[3-(1H-imidazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}pyridine
1-(3-chlorophenyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(oxan-4-yl)pyrimidin-2-amine
2-({2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)-6-methylquinolin-4-ol