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1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
4-benzyl-3-ethyl-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-1,4-diazepan-5-one
(3R,4S)-1-[3-(furan-2-yl)benzoyl]-4-propylpyrrolidin-3-amine
2-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}pyrrolidin-2-yl)-6-methyl-1H-1,3-benzodiazole
7-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[2-(dimethylamino)ethyl]-N-ethyl-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
3-[1-(2,5-dihydro-1H-pyrrole-2-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-4-amino-1-(4-chloro-1-methyl-1H-indole-2-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
3-[1-(5-ethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
(1S,5R)-3-(pyridine-2-carbonyl)-6-(pyrrolidine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[(5-methylthiophen-2-yl)methyl]propanamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-6-(piperidin-1-yl)pyrimidin-4-amine
N-methyl-N-(quinoxalin-2-ylmethyl)-4-sulfamoylbenzamide
ethyl 3,5-dimethyl-4-[3-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)piperidine-1-carbonyl]-1H-pyrrole-2-carboxylate
2-(phenoxymethyl)-8-[2-(thiophen-3-yl)acetyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-{1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})amine
4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2H-1,3-benzodioxole-5-carboxamide
N-[2-(4-sulfamoylphenyl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-[4-(dimethylamino)butanoyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
8-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4S)-1-(3-fluoropyridine-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-(4-fluoro-2-methylbenzenesulfonamido)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
(3R,4S)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-3,4-dimethylpiperidin-4-ol
1-{1-[2-(thiophen-2-yl)acetyl]piperidin-3-yl}pyrrolidin-2-one
2-ethoxy-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
3-[5-(1-benzylpiperidine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-cyclohexyl-4-[(dimethylamino)methyl]-N-(thiophen-3-ylmethyl)benzamide
N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3,5-dimethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-indole-2-carboxamide
6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(2-methoxyphenyl)ethyl]propanamide
5-(2,3-dihydro-1H-inden-1-ylmethyl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
(3R,7S,8aS)-7-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
methyl[(2E)-2-methylbut-2-en-1-yl]{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}piperidin-4-yl)methanesulfonamide
1-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-3-(propan-2-yl)urea
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(1-benzothiophen-2-ylmethyl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
1-{2-[1-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N3-(1-benzylpiperidin-4-yl)-N5-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-1-yl)pyridine-3-carboxamide
1-[4-(1H-imidazol-1-yl)benzoyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
methyl 3-[(3S,4R)-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl]propanoate
7-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]-1,2-dihydroisoquinolin-1-one
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(4-ethylphenyl)methyl]methylamine
(2E)-N-({3-methyl-7-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
1-(2-methoxy-5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol